WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | NEK1 | DIKSQNIFLTK | Lys2 | -6.9 | 1 | uM |
| WZ3105 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -2.1 | 1 | uM |
| WZ3105 | THP-1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | -9.0 | 1 | uM |
| WZ3105 | THP-1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -28.5 | 1 | uM |
| WZ3105 | THP-1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 50.1 | 1 | uM |
| WZ3105 | THP-1 | NEK9 | DIKTLNIFLTK | Lys2 | 13.2 | 1 | uM |
| WZ3105 | THP-1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 12.9 | 1 | uM |
| WZ3105 | THP-1 | MST1,MST2 | DIKAGNILLNTEGHAK | Lys2 | -3.3 | 1 | uM |
| WZ3105 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 35.1 | 1 | uM |
| WZ3105 | THP-1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 44.3 | 1 | uM |
| WZ3105 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -0.8 | 1 | uM |
| WZ3105 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -10.4 | 1 | uM |
| WZ3105 | THP-1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | -5.7 | 1 | uM |
| WZ3105 | THP-1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -12.9 | 1 | uM |
| WZ3105 | THP-1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -5.9 | 1 | uM |
| WZ3105 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | CDK13 | DIKCSNILLNNR | Lys2 | 26.6 | 1 | uM |
| WZ3105 | THP-1 | CDK9 | DMKAANVLITR | Lys2 | 23.4 | 1 | uM |
| WZ3105 | THP-1 | CDK16 | DLKPQNLLINER | Lys2 | 6.7 | 1 | uM |
| WZ3105 | THP-1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 6.5 | 1 | uM |
| WZ3105 | THP-1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 19.0 | 1 | uM |
| WZ3105 | THP-1 | PCTAIRE2 | DLKPQNLLINEK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | -12.3 | 1 | uM |
| WZ3105 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -11.4 | 1 | uM |
| WZ3105 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 0.6 | 1 | uM |