High-content imaging of six breast cancer cell lines treated with a library of small molecule kinase inhibitors. - Dataset (ID:20244)
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| Cell | SM Name | Small Mol Concentration | Small Mol Conc Unit | Other Reagent 1 Name | Other Reagent 1 Detection Channel | Other Reagent 2 Name | Other Reagent 2 Detection Channel | Row | Column | Field | X-coordinate | Y-coordinate | Image | Nuclear area (pixels) | Cytoplasm area (pixels) | Nuclear intensity (AU) | Std Dev of nuclear intensity (AU) | Cytoplasm intensity (AU) | Std Dev of cytoplasm intensity (AU) | 10% quantile of nuclear intensity (AU) | 20% quantile of nuclear intensity (AU) | 30% quantile of nuclear intensity (AU) | 40% quantile of nuclear intensity (AU) | 50% quantile of nuclear intensity (AU) | 60% quantile of nuclear intensity (AU) | 70% quantile of nuclear intensity (AU) | 80% quantile of nuclear intensity (AU) | 90% quantile of nuclear intensity (AU) | Ratio of cytoplasm perimeter to area | Cytoplasm perimeter (pixels) | Nuclear roundness | Nuclear length (pixels) | Nuclear halfwidth (pixels) | Number of nuclei | Ratio of nuclear perimeter to area | Nuclear perimeter (pixels) | Nuclear Haralick ASM | Nuclear Haralick contrast | Nuclear Haralick entropy | Nuclear Haralick IDM | Nuclear Haralick moment 2 | Nuclear Haralick moment 3 | Nuclear Haralick moment 4 | Nuclear Haralick moment 5 | Nuclear radial moment (border) | Nuclear radial moment (center) | Nuclear Threshold Adj Stat 1 (Threshold: 0.2) | Nuclear Threshold Adj Stat 1 (Threshold: 0.4) | Nuclear Threshold Adj Stat 2 (Threshold: 0.2) | Nuclear Threshold Adj Stat 2 (Threshold: 0.4) | Nuclear Threshold Adj Stat 3 (Threshold: 0.2) | Nuclear Threshold Adj Stat 3 (Threshold: 0.4) | Nuclear Threshold Adj Stat 4 (Threshold: 0.2) | Nuclear Threshold Adj Stat 4 (Threshold: 0.4) | Nuclear Threshold Adj Stat 5 (Threshold: 0.2) | Nuclear Threshold Adj Stat 5 (Threshold: 0.4) | Nuclear Threshold Adj Stat 6 (Threshold: 0.2) | Nuclear Threshold Adj Stat 6 (Threshold: 0.4) | Nuclear Threshold Adj Stat 7 (Threshold: 0.2) | Nuclear Threshold Adj Stat 7 (Threshold: 0.4) | Nuclear Threshold Adj Stat 8 (Threshold: 0.2) | Nuclear Threshold Adj Stat 8 (Threshold: 0.4) | Nuclear Threshold Adj Stat 9 (Threshold: 0.2) | Nuclear Threshold Adj Stat 9 (Threshold: 0.4) | Nuclear Threshold Adj Stat 10 (Threshold: 0.2) | Nuclear Threshold Adj Stat 10 (Threshold: 0.4) | Nuclear Threshold Adj Stat 11 (Threshold: 0.2) | Nuclear Threshold Adj Stat 11 (Threshold: 0.4) | Nuclear Threshold Adj Stat 12 (Threshold: 0.2) | Nuclear Threshold Adj Stat 12 (Threshold: 0.4) | Nuclear Threshold Adj Stat 13 (Threshold: 0.2) | Nuclear Threshold Adj Stat 13 (Threshold: 0.4) | Nuclear Threshold Adj Stat 14 (Threshold: 0.2) | Nuclear Threshold Adj Stat 14 (Threshold: 0.4) | Nuclear Threshold Adj Stat 15 (Threshold: 0.2) | Nuclear Threshold Adj Stat 15 (Threshold: 0.4) | Nuclear Threshold Adj Stat 16 (Threshold: 0.2) | Nuclear Threshold Adj Stat 16 (Threshold: 0.4) | Nuclear Threshold Adj Stat 17 (Threshold: 0.2) | Nuclear Threshold Adj Stat 17 (Threshold: 0.4) | Nuclear Threshold Adj Stat 18 (Threshold: 0.2) | Nuclear Threshold Adj Stat 18 (Threshold: 0.4) | Nuclear Threshold Adj Stat 19 (Threshold: 0.2) | Nuclear Threshold Adj Stat 19 (Threshold: 0.4) | Nuclear Threshold Adj Stat 20 (Threshold: 0.2) | Nuclear Threshold Adj Stat 20 (Threshold: 0.4) | Nuclear Threshold Adj Stat 21 (Threshold: 0.2) | Nuclear Threshold Adj Stat 21 (Threshold: 0.4) | Nuclear Threshold Adj Stat 22 (Threshold: 0.2) | Nuclear Threshold Adj Stat 22 (Threshold: 0.4) | Nuclear Threshold Adj Stat 23 (Threshold: 0.2) | Nuclear Threshold Adj Stat 23 (Threshold: 0.4) | Nuclear Threshold Adj Stat 24 (Threshold: 0.2) | Nuclear Threshold Adj Stat 24 (Threshold: 0.4) | Nuclear Threshold Adj Stat 25 (Threshold: 0.2) | Nuclear Threshold Adj Stat 25 (Threshold: 0.4) | Nuclear Threshold Adj Stat 26 (Threshold: 0.2) | Nuclear Threshold Adj Stat 26 (Threshold: 0.4) | Nuclear Threshold Adj Stat 27 (Threshold: 0.2) | Nuclear Threshold Adj Stat 27 (Threshold: 0.4) | Nuclear Threshold Adj Stat 28 | Nuclear Threshold Adj Stat 29 | Nuclear Threshold Adj Stat 30 | Nuclear Threshold Adj Stat 31 | Nuclear Threshold Adj Stat 32 | Nuclear Threshold Adj Stat 33 | Nuclear Threshold Adj Stat 34 | Nuclear Threshold Adj Stat 35 | Nuclear Threshold Adj Stat 36 | 10% quantile of cytoplasm intensity (AU) | 20% quantile of cytoplasm intensity (AU) | 30% quantile of cytoplasm intensity (AU) | 40% quantile of cytoplasm intensity (AU) | 50% quantile of cytoplasm intensity (AU) | 60% quantile of cytoplasm intensity (AU) | 70% quantile of cytoplasm intensity (AU) | 80% quantile of cytoplasm intensity (AU) | 90% quantile of cytoplasm intensity (AU) | Cytoplasmic Haralick ASM | Cytoplasmic Haralick contrast | Cytoplasmic Haralick entropy | Cytoplasmic Haralick IDM | Cytoplasmic Haralick moment 2 | Cytoplasmic Haralick moment 3 | Cytoplasmic Haralick moment 4 | Cytoplasmic Haralick moment 5 | Cytoplasmic radial moment (border) | Cytoplasmic radial moment (center) | Cytoplasmic Threshold Adj Stat 1 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 1 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 2 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 2 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 3 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 3 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 4 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 4 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 5 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 5 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 6 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 6 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 7 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 7 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 8 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 8 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 9 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 9 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 10 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 10 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 11 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 11 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 12 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 12 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 13 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 13 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 14 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 14 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 15 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 15 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 16 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 16 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 17 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 17 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 18 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 18 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 19 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 19 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 20 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 20 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 21 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 21 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 22 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 22 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 23 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 23 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 24 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 24 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 25 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 25 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 26 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 26 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 27 (Threshold: 0.2) | Cytoplasmic Threshold Adj Stat 27 (Threshold: 0.4) | Cytoplasmic Threshold Adj Stat 28 | Cytoplasmic Threshold Adj Stat 29 | Cytoplasmic Threshold Adj Stat 30 | Cytoplasmic Threshold Adj Stat 31 | Cytoplasmic Threshold Adj Stat 32 | Cytoplasmic Threshold Adj Stat 33 | Cytoplasmic Threshold Adj Stat 34 | Cytoplasmic Threshold Adj Stat 35 | Cytoplasmic Threshold Adj Stat 36 |
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| MDA-MB-231 | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 154 | 245 | | 7441 | 18098 | 595.1 | 99.87 | 158.05 | 276.24 | 459 | 515 | 549 | 576 | 598 | 618 | 640 | 669 | 725 | 0.0530 | 960 | 0.791 | 112.90 | 27.89 | 2 | 0.0372 | 277 | 0.0011 | 26.39 | 7.165 | 0.2288 | 364116.0 | 229000000 | 147000000000 | 96900000000000 | 0.4475 | 0.1984 | 0.0002 | 0.0000 | 0.0007 | 0.0001 | 0.0016 | 0.0000 | 0.0053 | 0.0005 | 0.0258 | 0.0124 | 0.0455 | 0.0206 | 0.0458 | 0.0151 | 0.0692 | 0.0230 | 0.8059 | 0.9282 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0002 | 0.0000 | 0.0020 | 0.0003 | 0.0163 | 0.0116 | 0.0267 | 0.0174 | 0.0252 | 0.0115 | 0.0358 | 0.0181 | 0.8938 | 0.9412 | 0.0093 | 0.0000 | 0.0093 | 0.0000 | 0.0093 | 0.0000 | 0.0292 | 0.0000 | 0.0560 | 0.0000 | 0.0840 | 0.0000 | 0.0793 | 0.0000 | 0.1039 | 0.0000 | 0.6196 | 0.0000 | 0.0018 | 0.0036 | 0.0094 | 0.0214 | 0.0420 | 0.0641 | 0.0646 | 0.0876 | 0.7055 | 11 | 14 | 17 | 20 | 25 | 35 | 85 | 239 | 575 | 0.1535 | 16.74 | 4.037 | 0.6476 | 101285.0 | 90600000 | 95000000000 | 112000000000000 | 0.3437 | 0.2785 | 0.0470 | 0.0020 | 0.1678 | 0.0214 | 0.1893 | 0.0935 | 0.1530 | 0.1136 | 0.1732 | 0.1877 | 0.0980 | 0.1717 | 0.0779 | 0.1236 | 0.0671 | 0.1142 | 0.0268 | 0.1723 | 0.0002 | 0.0000 | 0.0008 | 0.0002 | 0.0008 | 0.0013 | 0.0102 | 0.0086 | 0.0376 | 0.0335 | 0.0599 | 0.0539 | 0.0436 | 0.0392 | 0.0626 | 0.0588 | 0.7843 | 0.8046 | 0.0000 | 0.0003 | 0.0012 | 0.0000 | 0.0042 | 0.0040 | 0.0138 | 0.0138 | 0.0413 | 0.0458 | 0.0655 | 0.0684 | 0.0487 | 0.0468 | 0.0667 | 0.0620 | 0.7586 | 0.7589 | 0.0002 | 0.0007 | 0.0023 | 0.0114 | 0.0416 | 0.0654 | 0.0444 | 0.0633 | 0.7707 |
| MCF 10A | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 786 | 723 | | 4403 | 10505 | 156.8 | 37.21 | 158.32 | 156.07 | 111 | 125 | 136 | 145 | 154 | 163 | 173 | 187 | 207 | 0.0730 | 767 | 1.082 | 105.15 | 39.01 | 1 | 0.0620 | 273 | 0.0017 | 27.23 | 6.665 | 0.2280 | 25980.4 | 4530000 | 831000000 | 159000000000 | 0.4286 | 0.2358 | 0.0007 | 0.0000 | 0.0045 | 0.0003 | 0.0138 | 0.0018 | 0.0302 | 0.0040 | 0.0832 | 0.0260 | 0.1542 | 0.0510 | 0.1486 | 0.0545 | 0.1725 | 0.0808 | 0.3923 | 0.7817 | 0.0000 | 0.0000 | 0.0009 | 0.0002 | 0.0009 | 0.0002 | 0.0068 | 0.0009 | 0.0392 | 0.0176 | 0.0717 | 0.0309 | 0.0697 | 0.0248 | 0.0958 | 0.0405 | 0.7151 | 0.8849 | 0.0024 | 0.0182 | 0.0155 | 0.0146 | 0.0274 | 0.0474 | 0.0764 | 0.1314 | 0.1372 | 0.1788 | 0.2076 | 0.2336 | 0.1313 | 0.0985 | 0.1396 | 0.1314 | 0.2625 | 0.1460 | 0.0024 | 0.0015 | 0.0068 | 0.0336 | 0.0973 | 0.1357 | 0.1051 | 0.1367 | 0.4810 | 15 | 27 | 45 | 75 | 110 | 150 | 199 | 265 | 380 | 0.0051 | 65.67 | 6.760 | 0.3104 | 49420.1 | 21200000 | 11000000000 | 6460000000000 | 0.5076 | 0.1389 | 0.0172 | 0.0010 | 0.0968 | 0.0078 | 0.2177 | 0.0413 | 0.1765 | 0.0889 | 0.1820 | 0.1633 | 0.1360 | 0.1965 | 0.0859 | 0.1508 | 0.0522 | 0.1403 | 0.0357 | 0.2100 | 0.0006 | 0.0000 | 0.0015 | 0.0009 | 0.0038 | 0.0042 | 0.0125 | 0.0116 | 0.0563 | 0.0446 | 0.0987 | 0.0767 | 0.0747 | 0.0616 | 0.1081 | 0.0892 | 0.6439 | 0.7113 | 0.0009 | 0.0015 | 0.0030 | 0.0036 | 0.0093 | 0.0109 | 0.0246 | 0.0318 | 0.0818 | 0.0982 | 0.1325 | 0.1383 | 0.0971 | 0.0985 | 0.1250 | 0.1438 | 0.5259 | 0.4734 | 0.0002 | 0.0017 | 0.0057 | 0.0214 | 0.0664 | 0.1176 | 0.0927 | 0.1161 | 0.5782 | ||
| BT-20 | Barasertib | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 15 | 1 | 855 | 295 | | 10991 | 23655 | 262.5 | 76.92 | 158.35 | 201.26 | 177 | 198 | 216 | 232 | 250 | 269 | 292 | 321 | 366 | 0.0567 | 1341 | 1.156 | 118.61 | 44.10 | 2 | 0.0278 | 305 | 0.0005 | 81.23 | 7.822 | 0.1418 | 74835.2 | 23200000 | 7750000000 | 2800000000000 | 0.4804 | 0.1627 | 0.0002 | 0.0000 | 0.0011 | 0.0000 | 0.0071 | 0.0009 | 0.0294 | 0.0045 | 0.0907 | 0.0256 | 0.1763 | 0.0635 | 0.1516 | 0.0562 | 0.1834 | 0.0790 | 0.3603 | 0.7703 | 0.0000 | 0.0000 | 0.0004 | 0.0000 | 0.0012 | 0.0004 | 0.0117 | 0.0023 | 0.0349 | 0.0146 | 0.0759 | 0.0366 | 0.0625 | 0.0262 | 0.0909 | 0.0372 | 0.7224 | 0.8828 | 0.0004 | 0.0038 | 0.0059 | 0.0084 | 0.0143 | 0.0188 | 0.0412 | 0.0619 | 0.1017 | 0.1210 | 0.1509 | 0.1642 | 0.1076 | 0.1098 | 0.1366 | 0.1407 | 0.4414 | 0.3715 | 0.0008 | 0.0036 | 0.0096 | 0.0273 | 0.0644 | 0.1087 | 0.0818 | 0.1101 | 0.5937 | 10 | 12 | 15 | 20 | 43 | 109 | 209 | 323 | 476 | 0.0700 | 31.05 | 5.286 | 0.4973 | 65578.9 | 35100000 | 21700000000 | 15000000000000 | 0.5467 | 0.1326 | 0.0587 | 0.0020 | 0.2015 | 0.0205 | 0.3009 | 0.1523 | 0.1628 | 0.1523 | 0.1274 | 0.1764 | 0.0861 | 0.1946 | 0.0327 | 0.1099 | 0.0254 | 0.0900 | 0.0047 | 0.1020 | 0.0002 | 0.0002 | 0.0004 | 0.0001 | 0.0015 | 0.0005 | 0.0054 | 0.0054 | 0.0421 | 0.0359 | 0.0826 | 0.0761 | 0.0556 | 0.0480 | 0.0768 | 0.0648 | 0.7354 | 0.7690 | 0.0001 | 0.0000 | 0.0009 | 0.0009 | 0.0029 | 0.0031 | 0.0107 | 0.0130 | 0.0544 | 0.0570 | 0.1019 | 0.1180 | 0.0672 | 0.0698 | 0.0986 | 0.1004 | 0.6631 | 0.6377 | 0.0001 | 0.0002 | 0.0014 | 0.0079 | 0.0478 | 0.0936 | 0.0584 | 0.0901 | 0.7003 |
| MCF 10A | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 609 | 654 | | 7151 | 16942 | 197.2 | 47.67 | 158.72 | 128.62 | 142 | 158 | 169 | 180 | 191 | 204 | 217 | 235 | 262 | 0.0596 | 1009 | 1.165 | 114.14 | 40.26 | 1 | 0.0386 | 276 | 0.0010 | 44.53 | 7.179 | 0.1807 | 41154.1 | 9080000 | 2110000000 | 515000000000 | 0.4398 | 0.2146 | 0.0005 | 0.0000 | 0.0007 | 0.0000 | 0.0034 | 0.0005 | 0.0225 | 0.0016 | 0.0918 | 0.0226 | 0.1658 | 0.0544 | 0.1623 | 0.0541 | 0.1830 | 0.0721 | 0.3699 | 0.7947 | 0.0002 | 0.0000 | 0.0005 | 0.0000 | 0.0014 | 0.0003 | 0.0087 | 0.0007 | 0.0377 | 0.0140 | 0.0650 | 0.0283 | 0.0655 | 0.0241 | 0.0987 | 0.0339 | 0.7223 | 0.8987 | 0.0043 | 0.0021 | 0.0080 | 0.0062 | 0.0217 | 0.0331 | 0.0810 | 0.1198 | 0.1389 | 0.1818 | 0.1975 | 0.2293 | 0.1172 | 0.1198 | 0.1404 | 0.1446 | 0.2909 | 0.1632 | 0.0015 | 0.0028 | 0.0067 | 0.0294 | 0.0781 | 0.1246 | 0.1136 | 0.1476 | 0.4957 | 29 | 50 | 73 | 98 | 124 | 154 | 195 | 255 | 340 | 0.0025 | 49.37 | 6.896 | 0.3087 | 41734.7 | 14900000 | 6570000000 | 3430000000000 | 0.4757 | 0.1683 | 0.0102 | 0.0005 | 0.0551 | 0.0051 | 0.1533 | 0.0172 | 0.1688 | 0.0526 | 0.1754 | 0.1321 | 0.1767 | 0.1793 | 0.1141 | 0.1494 | 0.0913 | 0.1597 | 0.0551 | 0.3041 | 0.0000 | 0.0002 | 0.0006 | 0.0008 | 0.0042 | 0.0018 | 0.0120 | 0.0073 | 0.0502 | 0.0359 | 0.0871 | 0.0632 | 0.0784 | 0.0546 | 0.1087 | 0.0842 | 0.6587 | 0.7522 | 0.0021 | 0.0007 | 0.0015 | 0.0035 | 0.0069 | 0.0106 | 0.0218 | 0.0308 | 0.0832 | 0.0946 | 0.1321 | 0.1464 | 0.1017 | 0.1114 | 0.1388 | 0.1415 | 0.5118 | 0.4604 | 0.0011 | 0.0012 | 0.0050 | 0.0180 | 0.0637 | 0.1167 | 0.0942 | 0.1257 | 0.5744 | ||
| MCF 10A | Barasertib | 1.1 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 16 | 1 | 1116 | 643 | | 4192 | 3538 | 101.2 | 30.48 | 158.91 | 113.21 | 66 | 76 | 84 | 91 | 97 | 104 | 112 | 125 | 141 | 0.1888 | 668 | 0.252 | 105.39 | 16.55 | 4 | 0.1069 | 448 | 0.0013 | 39.51 | 6.913 | 0.1929 | 11171.4 | 1340000 | 175000000 | 24600000000 | 0.4594 | 0.2026 | 0.0014 | 0.0000 | 0.0041 | 0.0009 | 0.0124 | 0.0023 | 0.0464 | 0.0096 | 0.1319 | 0.0422 | 0.1994 | 0.0776 | 0.1641 | 0.0774 | 0.1567 | 0.1235 | 0.2835 | 0.6665 | 0.0006 | 0.0000 | 0.0010 | 0.0005 | 0.0022 | 0.0010 | 0.0128 | 0.0053 | 0.0491 | 0.0264 | 0.0952 | 0.0467 | 0.0789 | 0.0345 | 0.1084 | 0.0632 | 0.6518 | 0.8224 | 0.0000 | 0.0073 | 0.0032 | 0.0218 | 0.0170 | 0.0291 | 0.0668 | 0.1065 | 0.1188 | 0.1574 | 0.1739 | 0.1695 | 0.1294 | 0.1283 | 0.1379 | 0.1259 | 0.3531 | 0.2542 | 0.0016 | 0.0037 | 0.0132 | 0.0390 | 0.0895 | 0.1311 | 0.1101 | 0.1411 | 0.4708 | 37 | 66 | 88 | 111 | 133 | 160 | 195 | 241 | 311 | 0.0052 | 18.73 | 5.833 | 0.3641 | 38065.2 | 12000000 | 4640000000 | 2080000000000 | 0.5210 | 0.1303 | 0.0169 | 0.0013 | 0.0663 | 0.0074 | 0.1808 | 0.0207 | 0.1873 | 0.0702 | 0.1625 | 0.1318 | 0.1443 | 0.1839 | 0.0845 | 0.1498 | 0.0754 | 0.1639 | 0.0819 | 0.2709 | 0.0000 | 0.0000 | 0.0027 | 0.0009 | 0.0038 | 0.0021 | 0.0279 | 0.0141 | 0.0681 | 0.0513 | 0.1217 | 0.0881 | 0.1045 | 0.0783 | 0.1436 | 0.1245 | 0.5279 | 0.6407 | 0.0009 | 0.0047 | 0.0000 | 0.0107 | 0.0119 | 0.0225 | 0.0574 | 0.0664 | 0.1240 | 0.1163 | 0.1559 | 0.1720 | 0.1276 | 0.1139 | 0.1586 | 0.1649 | 0.3637 | 0.3286 | 0.0014 | 0.0028 | 0.0104 | 0.0369 | 0.0828 | 0.1711 | 0.1113 | 0.1474 | 0.4360 |
| MCF7 | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 803 | 843 | | 8078 | 37469 | 422.2 | 79.09 | 159.69 | 223.20 | 327 | 354 | 375 | 397 | 417 | 437 | 459 | 489 | 531 | 0.0317 | 1189 | 1.189 | 110.68 | 36.67 | 1 | 0.0326 | 263 | 0.0007 | 56.32 | 7.529 | 0.1530 | 184520.0 | 83400000 | 38900000000 | 18700000000000 | 0.4100 | 0.2411 | 0.0003 | 0.0000 | 0.0005 | 0.0000 | 0.0026 | 0.0001 | 0.0130 | 0.0004 | 0.0471 | 0.0139 | 0.1043 | 0.0293 | 0.1147 | 0.0226 | 0.1480 | 0.0455 | 0.5695 | 0.8882 | 0.0000 | 0.0000 | 0.0003 | 0.0000 | 0.0013 | 0.0000 | 0.0050 | 0.0000 | 0.0239 | 0.0107 | 0.0515 | 0.0209 | 0.0493 | 0.0112 | 0.0688 | 0.0227 | 0.8000 | 0.9344 | 0.0074 | 0.0206 | 0.0033 | 0.0155 | 0.0294 | 0.0722 | 0.0711 | 0.1598 | 0.1266 | 0.2268 | 0.1585 | 0.1701 | 0.1152 | 0.1495 | 0.1479 | 0.0979 | 0.3407 | 0.0876 | 0.0005 | 0.0054 | 0.0099 | 0.0311 | 0.0677 | 0.1022 | 0.1066 | 0.1196 | 0.5569 | 8 | 12 | 18 | 34 | 59 | 102 | 172 | 277 | 460 | 0.0551 | 26.43 | 5.339 | 0.4890 | 75319.8 | 53300000 | 47300000000 | 49000000000000 | 0.3610 | 0.2741 | 0.0647 | 0.0026 | 0.2087 | 0.0190 | 0.2734 | 0.1221 | 0.1568 | 0.1521 | 0.1237 | 0.2054 | 0.0877 | 0.1850 | 0.0465 | 0.1224 | 0.0270 | 0.0989 | 0.0115 | 0.0926 | 0.0006 | 0.0004 | 0.0007 | 0.0010 | 0.0031 | 0.0025 | 0.0146 | 0.0116 | 0.0594 | 0.0555 | 0.0986 | 0.0841 | 0.0693 | 0.0619 | 0.0969 | 0.0912 | 0.6568 | 0.6917 | 0.0009 | 0.0003 | 0.0015 | 0.0012 | 0.0039 | 0.0068 | 0.0169 | 0.0173 | 0.0767 | 0.0907 | 0.1116 | 0.1149 | 0.0824 | 0.0817 | 0.1129 | 0.1235 | 0.5932 | 0.5636 | 0.0006 | 0.0018 | 0.0039 | 0.0139 | 0.0709 | 0.1068 | 0.0718 | 0.1079 | 0.6224 |
| BT-20 | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 150 | 710 | | 6177 | 14509 | 257.7 | 49.98 | 159.94 | 175.38 | 195 | 216 | 230 | 243 | 255 | 267 | 280 | 296 | 323 | 0.0733 | 1064 | 0.993 | 123.79 | 34.53 | 1 | 0.0478 | 295 | 0.0009 | 53.18 | 7.248 | 0.1699 | 68920.1 | 19100000 | 5500000000 | 1640000000000 | 0.4318 | 0.2171 | 0.0000 | 0.0000 | 0.0009 | 0.0002 | 0.0030 | 0.0002 | 0.0173 | 0.0017 | 0.0536 | 0.0129 | 0.0983 | 0.0305 | 0.1154 | 0.0290 | 0.1599 | 0.0498 | 0.5517 | 0.8757 | 0.0000 | 0.0000 | 0.0004 | 0.0002 | 0.0013 | 0.0000 | 0.0044 | 0.0013 | 0.0238 | 0.0098 | 0.0441 | 0.0207 | 0.0492 | 0.0117 | 0.0819 | 0.0218 | 0.7949 | 0.9346 | 0.0103 | 0.0328 | 0.0091 | 0.0437 | 0.0343 | 0.1202 | 0.0926 | 0.1421 | 0.1669 | 0.1585 | 0.1829 | 0.1530 | 0.1291 | 0.0710 | 0.1451 | 0.1202 | 0.2297 | 0.1585 | 0.0007 | 0.0031 | 0.0099 | 0.0358 | 0.0782 | 0.1328 | 0.1171 | 0.1540 | 0.4684 | 16 | 20 | 33 | 57 | 93 | 139 | 201 | 286 | 409 | 0.0208 | 27.02 | 5.804 | 0.4346 | 56339.0 | 28300000 | 18000000000 | 13700000000000 | 0.5203 | 0.1387 | 0.0476 | 0.0018 | 0.1694 | 0.0111 | 0.2272 | 0.1026 | 0.1326 | 0.1244 | 0.1282 | 0.1647 | 0.1104 | 0.1591 | 0.0736 | 0.1121 | 0.0615 | 0.1069 | 0.0495 | 0.2172 | 0.0002 | 0.0000 | 0.0018 | 0.0007 | 0.0049 | 0.0018 | 0.0131 | 0.0102 | 0.0685 | 0.0529 | 0.1030 | 0.0883 | 0.0768 | 0.0614 | 0.1123 | 0.0986 | 0.6194 | 0.6860 | 0.0007 | 0.0003 | 0.0022 | 0.0038 | 0.0046 | 0.0082 | 0.0208 | 0.0260 | 0.0828 | 0.0984 | 0.1265 | 0.1386 | 0.0956 | 0.0989 | 0.1283 | 0.1435 | 0.5386 | 0.4824 | 0.0004 | 0.0027 | 0.0042 | 0.0175 | 0.0747 | 0.1189 | 0.0808 | 0.1256 | 0.5753 |
| MCF 10A | Barasertib | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 15 | 1 | 293 | 599 | | 8522 | 18731 | 124.8 | 36.07 | 159.94 | 131.22 | 85 | 96 | 104 | 111 | 119 | 128 | 138 | 151 | 171 | 0.0579 | 1085 | 0.655 | 121.63 | 30.46 | 3 | 0.0413 | 352 | 0.0021 | 21.46 | 6.543 | 0.2583 | 16874.9 | 2480000 | 397000000 | 69100000000 | 0.4218 | 0.2248 | 0.0015 | 0.0001 | 0.0032 | 0.0001 | 0.0107 | 0.0008 | 0.0379 | 0.0042 | 0.1011 | 0.0264 | 0.1598 | 0.0609 | 0.1590 | 0.0612 | 0.1920 | 0.0880 | 0.3347 | 0.7581 | 0.0008 | 0.0001 | 0.0009 | 0.0000 | 0.0028 | 0.0005 | 0.0110 | 0.0015 | 0.0388 | 0.0136 | 0.0711 | 0.0348 | 0.0644 | 0.0249 | 0.0950 | 0.0373 | 0.7152 | 0.8874 | 0.0062 | 0.0081 | 0.0090 | 0.0161 | 0.0225 | 0.0323 | 0.0749 | 0.0833 | 0.1256 | 0.1815 | 0.1532 | 0.1505 | 0.1256 | 0.1183 | 0.1369 | 0.1465 | 0.3459 | 0.2634 | 0.0016 | 0.0021 | 0.0083 | 0.0359 | 0.0826 | 0.1188 | 0.1038 | 0.1330 | 0.5139 | 17 | 35 | 65 | 98 | 134 | 170 | 212 | 264 | 339 | 0.0080 | 16.54 | 6.041 | 0.3804 | 42799.9 | 14800000 | 6050000000 | 2820000000000 | 0.4714 | 0.1684 | 0.0176 | 0.0010 | 0.0946 | 0.0066 | 0.2089 | 0.0387 | 0.1898 | 0.0857 | 0.1697 | 0.1579 | 0.1371 | 0.1913 | 0.0887 | 0.1635 | 0.0659 | 0.1531 | 0.0277 | 0.2022 | 0.0001 | 0.0001 | 0.0011 | 0.0005 | 0.0034 | 0.0022 | 0.0141 | 0.0087 | 0.0522 | 0.0394 | 0.0960 | 0.0745 | 0.0872 | 0.0648 | 0.1214 | 0.0920 | 0.6245 | 0.7178 | 0.0011 | 0.0016 | 0.0031 | 0.0070 | 0.0130 | 0.0169 | 0.0317 | 0.0396 | 0.0907 | 0.1065 | 0.1413 | 0.1568 | 0.1106 | 0.1168 | 0.1370 | 0.1456 | 0.4715 | 0.4093 | 0.0009 | 0.0021 | 0.0059 | 0.0218 | 0.0735 | 0.1242 | 0.1046 | 0.1292 | 0.5378 |
| MCF 10A | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 1086 | 620 | | 4452 | 3745 | 173.1 | 35.31 | 160.12 | 114.34 | 133 | 145 | 153 | 161 | 169 | 177 | 186 | 197 | 216 | 0.1522 | 570 | 1.194 | 77.34 | 28.86 | 1 | 0.0442 | 197 | 0.0021 | 21.97 | 6.469 | 0.2475 | 31225.1 | 5890000 | 1170000000 | 246000000000 | 0.3936 | 0.2497 | 0.0000 | 0.0000 | 0.0013 | 0.0000 | 0.0053 | 0.0002 | 0.0175 | 0.0012 | 0.0519 | 0.0169 | 0.1051 | 0.0386 | 0.1236 | 0.0286 | 0.1721 | 0.0435 | 0.5232 | 0.8710 | 0.0000 | 0.0000 | 0.0008 | 0.0000 | 0.0026 | 0.0002 | 0.0100 | 0.0009 | 0.0257 | 0.0133 | 0.0524 | 0.0252 | 0.0561 | 0.0137 | 0.0820 | 0.0252 | 0.7704 | 0.9216 | 0.0032 | 0.0056 | 0.0323 | 0.0113 | 0.0258 | 0.0339 | 0.0855 | 0.0734 | 0.1403 | 0.1864 | 0.1645 | 0.2034 | 0.1339 | 0.0847 | 0.1339 | 0.1073 | 0.2806 | 0.2938 | 0.0020 | 0.0039 | 0.0158 | 0.0331 | 0.0805 | 0.1051 | 0.1111 | 0.1362 | 0.5123 | 40 | 68 | 87 | 108 | 131 | 156 | 189 | 244 | 330 | 0.0027 | 39.04 | 6.449 | 0.3029 | 38710.2 | 12200000 | 4630000000 | 1970000000000 | 0.4732 | 0.1655 | 0.0072 | 0.0025 | 0.0929 | 0.0144 | 0.1158 | 0.0439 | 0.1411 | 0.0640 | 0.1496 | 0.1193 | 0.1604 | 0.1532 | 0.1086 | 0.1293 | 0.0989 | 0.1494 | 0.1255 | 0.3239 | 0.0021 | 0.0012 | 0.0031 | 0.0032 | 0.0093 | 0.0057 | 0.0260 | 0.0114 | 0.0639 | 0.0584 | 0.1070 | 0.0852 | 0.0826 | 0.0697 | 0.1158 | 0.1010 | 0.5903 | 0.6642 | 0.0027 | 0.0011 | 0.0046 | 0.0057 | 0.0146 | 0.0137 | 0.0401 | 0.0538 | 0.0866 | 0.0985 | 0.1486 | 0.1546 | 0.0902 | 0.1168 | 0.1395 | 0.1730 | 0.4731 | 0.3826 | 0.0021 | 0.0041 | 0.0110 | 0.0336 | 0.0782 | 0.1221 | 0.0912 | 0.1276 | 0.5302 |
| BT-20 | Barasertib | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 15 | 1 | 459 | 658 | | 11362 | 20851 | 286.6 | 57.22 | 160.43 | 166.77 | 216 | 238 | 254 | 268 | 283 | 297 | 315 | 335 | 362 | 0.0609 | 1269 | 1.250 | 84.58 | 36.89 | 1 | 0.0202 | 229 | 0.0006 | 69.33 | 7.619 | 0.1453 | 85435.4 | 26400000 | 8470000000 | 2810000000000 | 0.3998 | 0.2496 | 0.0001 | 0.0000 | 0.0008 | 0.0000 | 0.0026 | 0.0000 | 0.0151 | 0.0008 | 0.0564 | 0.0119 | 0.1324 | 0.0353 | 0.1449 | 0.0348 | 0.1680 | 0.0534 | 0.4798 | 0.8638 | 0.0001 | 0.0000 | 0.0005 | 0.0000 | 0.0011 | 0.0000 | 0.0057 | 0.0004 | 0.0244 | 0.0088 | 0.0561 | 0.0236 | 0.0596 | 0.0148 | 0.0768 | 0.0231 | 0.7756 | 0.9293 | 0.0061 | 0.0143 | 0.0094 | 0.0544 | 0.0304 | 0.0716 | 0.0839 | 0.1777 | 0.1733 | 0.2521 | 0.1926 | 0.1519 | 0.1291 | 0.0917 | 0.1512 | 0.0974 | 0.2241 | 0.0888 | 0.0015 | 0.0022 | 0.0078 | 0.0347 | 0.0806 | 0.1342 | 0.1129 | 0.1362 | 0.4899 | 14 | 18 | 28 | 51 | 95 | 156 | 222 | 299 | 405 | 0.0196 | 36.84 | 6.010 | 0.3723 | 53550.1 | 23300000 | 11800000000 | 6650000000000 | 0.5064 | 0.1481 | 0.0625 | 0.0012 | 0.2600 | 0.0157 | 0.3022 | 0.1503 | 0.1409 | 0.1993 | 0.0988 | 0.2074 | 0.0736 | 0.1703 | 0.0334 | 0.0942 | 0.0252 | 0.0818 | 0.0034 | 0.0799 | 0.0001 | 0.0000 | 0.0004 | 0.0005 | 0.0019 | 0.0015 | 0.0115 | 0.0099 | 0.0600 | 0.0532 | 0.1157 | 0.0968 | 0.0747 | 0.0636 | 0.1141 | 0.0984 | 0.6214 | 0.6761 | 0.0004 | 0.0010 | 0.0028 | 0.0037 | 0.0065 | 0.0110 | 0.0223 | 0.0260 | 0.0761 | 0.0864 | 0.1468 | 0.1528 | 0.0956 | 0.1004 | 0.1209 | 0.1293 | 0.5286 | 0.4895 | 0.0000 | 0.0010 | 0.0039 | 0.0157 | 0.0717 | 0.1279 | 0.0896 | 0.1188 | 0.5713 |
| MCF 10A | Barasertib | 1.1 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 16 | 1 | 84 | 350 | | 635 | 11961 | 63.2 | 10.04 | 161.70 | 197.63 | 50 | 54 | 57 | 61 | 63 | 66 | 68 | 71 | 76 | 0.0579 | 693 | 0.875 | 142.76 | 45.97 | 2 | 0.6299 | 400 | 0.0068 | 11.22 | 5.192 | 0.3174 | 4092.7 | 271580 | 18400000 | 1280000000 | 0.4246 | 0.2192 | 0.0020 | 0.0000 | 0.0061 | 0.0016 | 0.0242 | 0.0048 | 0.0364 | 0.0111 | 0.0667 | 0.0430 | 0.1091 | 0.0685 | 0.1172 | 0.0525 | 0.1960 | 0.0812 | 0.4424 | 0.7373 | 0.0018 | 0.0000 | 0.0053 | 0.0016 | 0.0124 | 0.0047 | 0.0284 | 0.0110 | 0.0443 | 0.0379 | 0.0585 | 0.0694 | 0.0709 | 0.0394 | 0.0816 | 0.0599 | 0.6968 | 0.7760 | 0.0580 | 0.3333 | 0.0870 | 0.0000 | 0.1594 | 0.3333 | 0.0725 | 0.3333 | 0.1739 | 0.0000 | 0.0870 | 0.0000 | 0.0580 | 0.0000 | 0.1014 | 0.0000 | 0.2029 | 0.0000 | 0.0060 | 0.0030 | 0.0328 | 0.0448 | 0.0836 | 0.1045 | 0.1104 | 0.1761 | 0.4388 | 14 | 18 | 22 | 31 | 58 | 116 | 205 | 315 | 458 | 0.0352 | 28.43 | 5.403 | 0.4619 | 65200.6 | 35400000 | 22500000000 | 16100000000000 | 0.5927 | 0.1032 | 0.1018 | 0.0034 | 0.2284 | 0.0353 | 0.3243 | 0.1826 | 0.1467 | 0.1894 | 0.1089 | 0.2031 | 0.0462 | 0.1570 | 0.0249 | 0.0990 | 0.0130 | 0.0728 | 0.0059 | 0.0575 | 0.0002 | 0.0000 | 0.0009 | 0.0004 | 0.0020 | 0.0022 | 0.0142 | 0.0124 | 0.0583 | 0.0519 | 0.0965 | 0.0944 | 0.0720 | 0.0609 | 0.0991 | 0.0924 | 0.6569 | 0.6855 | 0.0000 | 0.0000 | 0.0016 | 0.0006 | 0.0029 | 0.0060 | 0.0195 | 0.0279 | 0.0776 | 0.0835 | 0.1193 | 0.1370 | 0.0921 | 0.0943 | 0.1271 | 0.1346 | 0.5598 | 0.5161 | 0.0002 | 0.0002 | 0.0027 | 0.0176 | 0.0677 | 0.1015 | 0.0832 | 0.1135 | 0.6134 |
| Hs 578T | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 324 | 200 | | 9267 | 28546 | 136.9 | 41.75 | 161.87 | 233.98 | 86 | 99 | 112 | 124 | 135 | 146 | 158 | 172 | 193 | 0.0455 | 1300 | 0.914 | 69.01 | 19.70 | 6 | 0.0181 | 168 | 0.0013 | 24.49 | 6.895 | 0.2332 | 20479.4 | 3300000 | 567000000 | 103000000000 | 0.4196 | 0.2164 | 0.0018 | 0.0000 | 0.0058 | 0.0004 | 0.0076 | 0.0017 | 0.0306 | 0.0073 | 0.1008 | 0.0279 | 0.1517 | 0.0559 | 0.1639 | 0.0691 | 0.1899 | 0.0994 | 0.3480 | 0.7382 | 0.0006 | 0.0000 | 0.0024 | 0.0000 | 0.0018 | 0.0004 | 0.0088 | 0.0035 | 0.0321 | 0.0139 | 0.0490 | 0.0251 | 0.0522 | 0.0285 | 0.0722 | 0.0388 | 0.7809 | 0.8897 | 0.0043 | 0.0081 | 0.0086 | 0.0070 | 0.0241 | 0.0252 | 0.0455 | 0.0916 | 0.0769 | 0.1370 | 0.1327 | 0.1631 | 0.1078 | 0.1269 | 0.1430 | 0.1511 | 0.4570 | 0.2900 | 0.0011 | 0.0051 | 0.0058 | 0.0210 | 0.0568 | 0.0917 | 0.0790 | 0.1085 | 0.6310 | 20 | 25 | 32 | 42 | 59 | 88 | 146 | 248 | 465 | 0.0337 | 41.47 | 5.283 | 0.5159 | 80948.0 | 65000000 | 65600000000 | 76000000000000 | 0.5258 | 0.1466 | 0.0551 | 0.0017 | 0.1968 | 0.0211 | 0.2532 | 0.1230 | 0.1516 | 0.1351 | 0.1376 | 0.1940 | 0.0880 | 0.1858 | 0.0596 | 0.1152 | 0.0384 | 0.1031 | 0.0199 | 0.1210 | 0.0003 | 0.0001 | 0.0003 | 0.0004 | 0.0036 | 0.0018 | 0.0190 | 0.0156 | 0.0709 | 0.0590 | 0.1046 | 0.0925 | 0.0709 | 0.0629 | 0.1037 | 0.0968 | 0.6266 | 0.6709 | 0.0006 | 0.0008 | 0.0014 | 0.0019 | 0.0072 | 0.0074 | 0.0231 | 0.0271 | 0.0831 | 0.0907 | 0.1334 | 0.1460 | 0.0842 | 0.0925 | 0.1238 | 0.1209 | 0.5433 | 0.5125 | 0.0008 | 0.0026 | 0.0043 | 0.0227 | 0.0776 | 0.1148 | 0.0780 | 0.1182 | 0.5810 |
| Hs 578T | Barasertib | 10 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 15 | 1 | 207 | 478 | | 13048 | 26519 | 97.0 | 27.99 | 161.98 | 234.77 | 64 | 74 | 81 | 88 | 95 | 102 | 109 | 119 | 134 | 0.0514 | 1363 | 0.414 | 318.40 | 44.82 | 2 | 0.0676 | 882 | 0.0022 | 19.38 | 6.429 | 0.2488 | 10191.1 | 1150000 | 139000000 | 17800000000 | 0.4486 | 0.1898 | 0.0006 | 0.0001 | 0.0026 | 0.0001 | 0.0142 | 0.0005 | 0.0573 | 0.0057 | 0.1294 | 0.0245 | 0.1873 | 0.0596 | 0.1931 | 0.0819 | 0.1988 | 0.1265 | 0.2168 | 0.7010 | 0.0000 | 0.0000 | 0.0002 | 0.0000 | 0.0021 | 0.0002 | 0.0123 | 0.0021 | 0.0425 | 0.0125 | 0.0796 | 0.0275 | 0.0907 | 0.0335 | 0.1311 | 0.0529 | 0.6415 | 0.8713 | 0.0086 | 0.0180 | 0.0124 | 0.0237 | 0.0341 | 0.0606 | 0.0834 | 0.1219 | 0.1405 | 0.1457 | 0.1777 | 0.1833 | 0.1230 | 0.1129 | 0.1467 | 0.1211 | 0.2735 | 0.2128 | 0.0013 | 0.0034 | 0.0092 | 0.0433 | 0.0938 | 0.1445 | 0.1259 | 0.1491 | 0.4295 | 12 | 14 | 16 | 18 | 33 | 81 | 172 | 311 | 501 | 0.1539 | 30.24 | 4.603 | 0.5818 | 81353.0 | 57600000 | 49500000000 | 48800000000000 | 0.6313 | 0.0832 | 0.0968 | 0.0061 | 0.2891 | 0.0382 | 0.3119 | 0.2073 | 0.1514 | 0.1858 | 0.0786 | 0.1931 | 0.0396 | 0.1633 | 0.0221 | 0.0966 | 0.0084 | 0.0664 | 0.0019 | 0.0433 | 0.0002 | 0.0001 | 0.0014 | 0.0006 | 0.0029 | 0.0019 | 0.0159 | 0.0126 | 0.0664 | 0.0555 | 0.1013 | 0.0925 | 0.0752 | 0.0680 | 0.1062 | 0.0957 | 0.6305 | 0.6731 | 0.0001 | 0.0004 | 0.0027 | 0.0026 | 0.0041 | 0.0069 | 0.0213 | 0.0238 | 0.0829 | 0.0859 | 0.1261 | 0.1347 | 0.0905 | 0.1014 | 0.1246 | 0.1340 | 0.5478 | 0.5103 | 0.0002 | 0.0021 | 0.0035 | 0.0166 | 0.0752 | 0.1103 | 0.0892 | 0.1185 | 0.5844 |
| BT-20 | Barasertib | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 15 | 1 | 634 | 836 | | 6694 | 23123 | 220.1 | 45.92 | 161.99 | 175.74 | 165 | 181 | 193 | 204 | 215 | 227 | 240 | 256 | 280 | 0.0480 | 1111 | 1.210 | 102.65 | 44.29 | 1 | 0.0420 | 281 | 0.0011 | 40.91 | 7.097 | 0.1838 | 50535.0 | 12100000 | 3040000000 | 797000000000 | 0.4401 | 0.2135 | 0.0002 | 0.0000 | 0.0007 | 0.0000 | 0.0029 | 0.0002 | 0.0159 | 0.0003 | 0.0615 | 0.0172 | 0.1197 | 0.0311 | 0.1488 | 0.0369 | 0.1834 | 0.0515 | 0.4669 | 0.8628 | 0.0000 | 0.0000 | 0.0002 | 0.0000 | 0.0014 | 0.0000 | 0.0062 | 0.0000 | 0.0277 | 0.0126 | 0.0551 | 0.0171 | 0.0627 | 0.0163 | 0.0885 | 0.0249 | 0.7582 | 0.9291 | 0.0046 | 0.0108 | 0.0147 | 0.0179 | 0.0394 | 0.0502 | 0.0879 | 0.1613 | 0.1319 | 0.1613 | 0.1712 | 0.1864 | 0.1071 | 0.1111 | 0.1328 | 0.0932 | 0.3104 | 0.2079 | 0.0013 | 0.0016 | 0.0090 | 0.0303 | 0.0940 | 0.1211 | 0.1137 | 0.1523 | 0.4767 | 11 | 13 | 18 | 38 | 92 | 162 | 235 | 308 | 417 | 0.0450 | 24.09 | 5.615 | 0.4490 | 57122.6 | 25900000 | 13700000000 | 8060000000000 | 0.4415 | 0.1960 | 0.0450 | 0.0017 | 0.1921 | 0.0096 | 0.3192 | 0.0939 | 0.1711 | 0.1707 | 0.1124 | 0.2071 | 0.0816 | 0.1996 | 0.0401 | 0.1194 | 0.0308 | 0.1084 | 0.0078 | 0.0896 | 0.0005 | 0.0001 | 0.0009 | 0.0005 | 0.0008 | 0.0016 | 0.0092 | 0.0074 | 0.0453 | 0.0386 | 0.0833 | 0.0715 | 0.0621 | 0.0516 | 0.0918 | 0.0767 | 0.7061 | 0.7520 | 0.0001 | 0.0007 | 0.0010 | 0.0017 | 0.0034 | 0.0074 | 0.0198 | 0.0214 | 0.0603 | 0.0717 | 0.1056 | 0.1113 | 0.0810 | 0.0864 | 0.1068 | 0.1131 | 0.6220 | 0.5862 | 0.0001 | 0.0006 | 0.0018 | 0.0130 | 0.0555 | 0.0911 | 0.0731 | 0.1019 | 0.6628 |
| MCF 10A | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 1013 | 776 | | 4132 | 4149 | 163.6 | 45.21 | 162.20 | 159.12 | 116 | 127 | 136 | 145 | 155 | 166 | 178 | 197 | 224 | 0.1347 | 559 | 1.127 | 94.07 | 29.83 | 1 | 0.0549 | 227 | 0.0016 | 35.59 | 6.765 | 0.2144 | 28795.0 | 5490000 | 1140000000 | 256000000000 | 0.3736 | 0.2711 | 0.0000 | 0.0000 | 0.0013 | 0.0000 | 0.0097 | 0.0000 | 0.0313 | 0.0016 | 0.1031 | 0.0289 | 0.1793 | 0.0586 | 0.1696 | 0.0559 | 0.1608 | 0.0805 | 0.3449 | 0.7744 | 0.0000 | 0.0000 | 0.0006 | 0.0000 | 0.0029 | 0.0000 | 0.0126 | 0.0012 | 0.0426 | 0.0173 | 0.0765 | 0.0318 | 0.0726 | 0.0202 | 0.0833 | 0.0333 | 0.7089 | 0.8961 | 0.0012 | 0.0057 | 0.0060 | 0.0028 | 0.0193 | 0.0342 | 0.0712 | 0.1026 | 0.1351 | 0.1852 | 0.1689 | 0.1538 | 0.1074 | 0.1254 | 0.1544 | 0.1282 | 0.3366 | 0.2621 | 0.0006 | 0.0029 | 0.0081 | 0.0400 | 0.0737 | 0.1398 | 0.0986 | 0.1119 | 0.5244 | 19 | 39 | 59 | 79 | 105 | 140 | 187 | 267 | 405 | 0.0058 | 51.95 | 6.395 | 0.3274 | 51621.9 | 23000000 | 12200000000 | 7280000000000 | 0.4555 | 0.1933 | 0.0214 | 0.0008 | 0.1246 | 0.0084 | 0.2206 | 0.0489 | 0.1851 | 0.1281 | 0.1495 | 0.1778 | 0.1388 | 0.1912 | 0.0747 | 0.1272 | 0.0534 | 0.1348 | 0.0320 | 0.1828 | 0.0006 | 0.0000 | 0.0011 | 0.0036 | 0.0034 | 0.0027 | 0.0238 | 0.0173 | 0.0747 | 0.0600 | 0.1065 | 0.1055 | 0.0821 | 0.0673 | 0.1121 | 0.1014 | 0.5957 | 0.6421 | 0.0017 | 0.0000 | 0.0033 | 0.0040 | 0.0083 | 0.0049 | 0.0282 | 0.0346 | 0.0698 | 0.0949 | 0.1412 | 0.1215 | 0.0947 | 0.1057 | 0.1204 | 0.1364 | 0.5324 | 0.4980 | 0.0007 | 0.0034 | 0.0103 | 0.0248 | 0.0765 | 0.1254 | 0.0827 | 0.1158 | 0.5603 |
| BT-20 | A443654 | 1.1 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 12 | 1 | 739 | 828 | | 3336 | 10996 | 733.4 | 131.67 | 162.29 | 302.51 | 560 | 619 | 661 | 696 | 729 | 766 | 805 | 848 | 907 | 0.0851 | 936 | 1.020 | 70.01 | 22.36 | 1 | 0.0525 | 175 | 0.0011 | 45.93 | 7.024 | 0.1864 | 555153.0 | 433000000 | 346000000000 | 284000000000000 | 0.4491 | 0.1924 | 0.0000 | 0.0000 | 0.0004 | 0.0000 | 0.0008 | 0.0000 | 0.0070 | 0.0003 | 0.0488 | 0.0168 | 0.1141 | 0.0324 | 0.0930 | 0.0251 | 0.1439 | 0.0321 | 0.5920 | 0.8934 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0024 | 0.0003 | 0.0255 | 0.0157 | 0.0541 | 0.0275 | 0.0375 | 0.0151 | 0.0620 | 0.0236 | 0.8185 | 0.9178 | 0.0041 | 0.0000 | 0.0000 | 0.0541 | 0.0269 | 0.1081 | 0.0579 | 0.2432 | 0.1467 | 0.1892 | 0.2004 | 0.2973 | 0.1240 | 0.0270 | 0.1508 | 0.0541 | 0.2893 | 0.0270 | 0.0000 | 0.0025 | 0.0105 | 0.0215 | 0.0732 | 0.0942 | 0.0905 | 0.1046 | 0.6031 | 8 | 10 | 11 | 12 | 14 | 20 | 71 | 262 | 593 | 0.2612 | 53.14 | 3.819 | 0.6522 | 117840.0 | 116000000 | 132000000000 | 164000000000000 | 0.5865 | 0.0859 | 0.1144 | 0.0083 | 0.2779 | 0.0904 | 0.2861 | 0.2629 | 0.1417 | 0.1599 | 0.1063 | 0.1460 | 0.0436 | 0.1252 | 0.0272 | 0.0918 | 0.0027 | 0.0668 | 0.0000 | 0.0487 | 0.0000 | 0.0000 | 0.0007 | 0.0003 | 0.0007 | 0.0007 | 0.0093 | 0.0101 | 0.0593 | 0.0520 | 0.1052 | 0.1002 | 0.0576 | 0.0598 | 0.1014 | 0.0881 | 0.6657 | 0.6888 | 0.0000 | 0.0008 | 0.0008 | 0.0013 | 0.0024 | 0.0051 | 0.0154 | 0.0166 | 0.0675 | 0.0696 | 0.1110 | 0.1099 | 0.0667 | 0.0743 | 0.1082 | 0.1002 | 0.6280 | 0.6222 | 0.0000 | 0.0007 | 0.0011 | 0.0136 | 0.0618 | 0.1045 | 0.0674 | 0.0986 | 0.6522 |
| MCF 10A | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 324 | 442 | | 5445 | 9682 | 138.7 | 35.79 | 163.09 | 136.98 | 98 | 109 | 117 | 125 | 133 | 142 | 152 | 165 | 188 | 0.0876 | 848 | 1.068 | 95.72 | 31.26 | 1 | 0.0455 | 248 | 0.0019 | 26.13 | 6.600 | 0.2423 | 20529.1 | 3240000 | 545000000 | 97400000000 | 0.4118 | 0.2366 | 0.0003 | 0.0000 | 0.0022 | 0.0000 | 0.0119 | 0.0004 | 0.0372 | 0.0029 | 0.0985 | 0.0264 | 0.1691 | 0.0554 | 0.1649 | 0.0532 | 0.1854 | 0.0975 | 0.3304 | 0.7642 | 0.0002 | 0.0000 | 0.0007 | 0.0000 | 0.0034 | 0.0000 | 0.0149 | 0.0009 | 0.0434 | 0.0150 | 0.0739 | 0.0264 | 0.0730 | 0.0186 | 0.1034 | 0.0390 | 0.6871 | 0.9000 | 0.0057 | 0.0136 | 0.0086 | 0.0181 | 0.0114 | 0.0317 | 0.0762 | 0.1134 | 0.1495 | 0.1950 | 0.1733 | 0.2109 | 0.1343 | 0.1293 | 0.1476 | 0.1383 | 0.2933 | 0.1497 | 0.0017 | 0.0033 | 0.0130 | 0.0401 | 0.0794 | 0.1216 | 0.1057 | 0.1358 | 0.4994 | 19 | 42 | 68 | 95 | 129 | 166 | 213 | 270 | 358 | 0.0040 | 66.08 | 6.940 | 0.2888 | 45362.2 | 16600000 | 7290000000 | 3700000000000 | 0.5293 | 0.1340 | 0.0265 | 0.0026 | 0.1297 | 0.0115 | 0.2310 | 0.0590 | 0.1394 | 0.1144 | 0.1490 | 0.1576 | 0.1355 | 0.1769 | 0.0839 | 0.1439 | 0.0606 | 0.1362 | 0.0445 | 0.1980 | 0.0006 | 0.0004 | 0.0010 | 0.0018 | 0.0023 | 0.0033 | 0.0177 | 0.0117 | 0.0586 | 0.0526 | 0.1291 | 0.0966 | 0.0780 | 0.0741 | 0.1126 | 0.0990 | 0.5999 | 0.6605 | 0.0015 | 0.0019 | 0.0018 | 0.0054 | 0.0111 | 0.0151 | 0.0348 | 0.0414 | 0.0860 | 0.1056 | 0.1631 | 0.1698 | 0.1002 | 0.0928 | 0.1236 | 0.1381 | 0.4778 | 0.4298 | 0.0010 | 0.0018 | 0.0061 | 0.0244 | 0.0786 | 0.1389 | 0.0972 | 0.1322 | 0.5198 | ||
| MCF7 | A443654 | 1.1 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 12 | 1 | 1271 | 351 | | 4157 | 9898 | 475.9 | 89.44 | 163.26 | 251.77 | 360 | 394 | 423 | 449 | 475 | 498 | 524 | 554 | 594 | 0.0813 | 805 | 1.028 | 152.20 | 40.79 | 2 | 0.0871 | 362 | 0.0008 | 73.60 | 7.318 | 0.1483 | 234454.0 | 119000000 | 62600000000 | 33700000000000 | 0.4174 | 0.2233 | 0.0003 | 0.0000 | 0.0010 | 0.0000 | 0.0017 | 0.0000 | 0.0196 | 0.0010 | 0.0716 | 0.0187 | 0.1191 | 0.0382 | 0.1160 | 0.0296 | 0.1725 | 0.0500 | 0.4981 | 0.8625 | 0.0003 | 0.0000 | 0.0003 | 0.0000 | 0.0009 | 0.0000 | 0.0069 | 0.0007 | 0.0343 | 0.0162 | 0.0480 | 0.0300 | 0.0474 | 0.0157 | 0.0809 | 0.0288 | 0.7811 | 0.9086 | 0.0000 | 0.0390 | 0.0204 | 0.0260 | 0.0471 | 0.1429 | 0.0973 | 0.2597 | 0.1476 | 0.2338 | 0.2057 | 0.1558 | 0.1350 | 0.0779 | 0.1162 | 0.0519 | 0.2308 | 0.0130 | 0.0010 | 0.0010 | 0.0048 | 0.0299 | 0.0676 | 0.1356 | 0.1236 | 0.1472 | 0.4894 | 7 | 10 | 13 | 22 | 39 | 75 | 136 | 293 | 547 | 0.0676 | 32.18 | 4.895 | 0.5343 | 90034.8 | 69000000 | 62100000000 | 62700000000000 | 0.5861 | 0.0893 | 0.0409 | 0.0025 | 0.1595 | 0.0187 | 0.2704 | 0.0934 | 0.2179 | 0.1214 | 0.1595 | 0.1766 | 0.0914 | 0.2054 | 0.0311 | 0.1350 | 0.0214 | 0.1180 | 0.0078 | 0.1290 | 0.0003 | 0.0003 | 0.0013 | 0.0017 | 0.0043 | 0.0049 | 0.0140 | 0.0129 | 0.0478 | 0.0466 | 0.0870 | 0.0765 | 0.0558 | 0.0552 | 0.0797 | 0.0797 | 0.7096 | 0.7222 | 0.0004 | 0.0000 | 0.0016 | 0.0017 | 0.0028 | 0.0043 | 0.0172 | 0.0170 | 0.0537 | 0.0679 | 0.1034 | 0.0909 | 0.0577 | 0.0635 | 0.0885 | 0.0905 | 0.6747 | 0.6642 | 0.0000 | 0.0026 | 0.0026 | 0.0125 | 0.0521 | 0.0922 | 0.0558 | 0.0845 | 0.6978 |
| BT-20 | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 357 | 710 | | 4921 | 10409 | 582.7 | 104.04 | 163.34 | 169.37 | 446 | 495 | 525 | 552 | 579 | 603 | 634 | 667 | 722 | 0.0790 | 822 | 1.185 | 96.46 | 39.82 | 1 | 0.0528 | 260 | 0.0007 | 60.83 | 7.459 | 0.1592 | 350308.0 | 217000000 | 138000000000 | 90400000000000 | 0.4237 | 0.2197 | 0.0000 | 0.0000 | 0.0008 | 0.0000 | 0.0017 | 0.0004 | 0.0084 | 0.0015 | 0.0427 | 0.0174 | 0.0858 | 0.0245 | 0.0936 | 0.0272 | 0.1375 | 0.0367 | 0.6295 | 0.8923 | 0.0000 | 0.0000 | 0.0002 | 0.0000 | 0.0007 | 0.0000 | 0.0031 | 0.0002 | 0.0252 | 0.0151 | 0.0417 | 0.0191 | 0.0370 | 0.0165 | 0.0620 | 0.0242 | 0.8301 | 0.9248 | 0.0075 | 0.0326 | 0.0090 | 0.0000 | 0.0271 | 0.0761 | 0.0827 | 0.1739 | 0.1203 | 0.1739 | 0.1399 | 0.2391 | 0.1068 | 0.1413 | 0.1053 | 0.1087 | 0.4015 | 0.0543 | 0.0017 | 0.0034 | 0.0029 | 0.0253 | 0.0623 | 0.1077 | 0.1098 | 0.1355 | 0.5513 | 11 | 14 | 21 | 52 | 104 | 160 | 229 | 315 | 422 | 0.0230 | 43.80 | 6.033 | 0.3963 | 55363.2 | 23600000 | 11400000000 | 6020000000000 | 0.5634 | 0.1337 | 0.0386 | 0.0005 | 0.1929 | 0.0101 | 0.2671 | 0.0648 | 0.1977 | 0.1411 | 0.1244 | 0.2046 | 0.0839 | 0.1945 | 0.0473 | 0.1177 | 0.0260 | 0.1172 | 0.0222 | 0.1494 | 0.0000 | 0.0002 | 0.0002 | 0.0006 | 0.0024 | 0.0004 | 0.0120 | 0.0066 | 0.0468 | 0.0368 | 0.0843 | 0.0643 | 0.0646 | 0.0509 | 0.1058 | 0.0885 | 0.6839 | 0.7518 | 0.0008 | 0.0003 | 0.0011 | 0.0016 | 0.0036 | 0.0038 | 0.0149 | 0.0166 | 0.0618 | 0.0787 | 0.1118 | 0.1234 | 0.0845 | 0.0918 | 0.1220 | 0.1321 | 0.5995 | 0.5516 | 0.0005 | 0.0010 | 0.0027 | 0.0124 | 0.0553 | 0.0981 | 0.0694 | 0.1131 | 0.6476 | ||
| BT-20 | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 219 | 745 | | 5417 | 7682 | 459.9 | 105.22 | 163.49 | 154.87 | 337 | 370 | 397 | 421 | 446 | 473 | 502 | 541 | 606 | 0.1009 | 775 | 0.952 | 103.82 | 28.00 | 1 | 0.0462 | 250 | 0.0007 | 65.25 | 7.472 | 0.1512 | 222541.0 | 113000000 | 60600000000 | 34000000000000 | 0.4352 | 0.2219 | 0.0006 | 0.0000 | 0.0009 | 0.0002 | 0.0012 | 0.0002 | 0.0160 | 0.0018 | 0.0690 | 0.0207 | 0.1406 | 0.0417 | 0.1432 | 0.0435 | 0.1788 | 0.0688 | 0.4498 | 0.8231 | 0.0005 | 0.0000 | 0.0002 | 0.0000 | 0.0005 | 0.0000 | 0.0073 | 0.0006 | 0.0381 | 0.0131 | 0.0709 | 0.0252 | 0.0628 | 0.0204 | 0.0986 | 0.0385 | 0.7212 | 0.9023 | 0.0061 | 0.0059 | 0.0163 | 0.0088 | 0.0132 | 0.0147 | 0.0499 | 0.1003 | 0.0957 | 0.1504 | 0.1232 | 0.1681 | 0.0896 | 0.1386 | 0.0998 | 0.1534 | 0.5061 | 0.2596 | 0.0016 | 0.0041 | 0.0086 | 0.0345 | 0.0858 | 0.1248 | 0.0998 | 0.1281 | 0.5127 | 16 | 24 | 47 | 80 | 120 | 162 | 209 | 275 | 401 | 0.0119 | 39.04 | 6.336 | 0.3337 | 50710.0 | 20800000 | 10000000000 | 5380000000000 | 0.5608 | 0.1109 | 0.0360 | 0.0009 | 0.1274 | 0.0147 | 0.1801 | 0.0477 | 0.1670 | 0.1198 | 0.1511 | 0.1590 | 0.1292 | 0.1862 | 0.1002 | 0.1203 | 0.0712 | 0.1323 | 0.0378 | 0.2192 | 0.0008 | 0.0002 | 0.0011 | 0.0005 | 0.0016 | 0.0021 | 0.0153 | 0.0143 | 0.0629 | 0.0509 | 0.1018 | 0.0835 | 0.0862 | 0.0685 | 0.1314 | 0.1042 | 0.5988 | 0.6757 | 0.0020 | 0.0020 | 0.0016 | 0.0045 | 0.0115 | 0.0109 | 0.0262 | 0.0377 | 0.0994 | 0.0942 | 0.1224 | 0.1413 | 0.0970 | 0.0932 | 0.1431 | 0.1413 | 0.4968 | 0.4750 | 0.0000 | 0.0010 | 0.0056 | 0.0203 | 0.0811 | 0.1353 | 0.0889 | 0.1366 | 0.5312 | ||
| BT-20 | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 213 | 896 | | 3746 | 14440 | 324.0 | 67.68 | 163.52 | 174.35 | 235 | 267 | 288 | 305 | 322 | 340 | 359 | 382 | 414 | 0.0614 | 886 | 1.026 | 90.35 | 31.58 | 1 | 0.0670 | 251 | 0.0007 | 89.85 | 7.502 | 0.1378 | 109544.0 | 38500000 | 14000000000 | 5270000000000 | 0.4313 | 0.2081 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0025 | 0.0008 | 0.0143 | 0.0014 | 0.0573 | 0.0161 | 0.1297 | 0.0417 | 0.1481 | 0.0296 | 0.1661 | 0.0735 | 0.4822 | 0.8369 | 0.0000 | 0.0000 | 0.0000 | 0.0000 | 0.0006 | 0.0005 | 0.0052 | 0.0014 | 0.0223 | 0.0128 | 0.0419 | 0.0312 | 0.0461 | 0.0115 | 0.0652 | 0.0325 | 0.8187 | 0.9101 | 0.0015 | 0.0741 | 0.0092 | 0.0556 | 0.0382 | 0.0926 | 0.0947 | 0.1667 | 0.1740 | 0.1852 | 0.1969 | 0.1481 | 0.1191 | 0.0926 | 0.1481 | 0.1111 | 0.2183 | 0.0741 | 0.0000 | 0.0005 | 0.0054 | 0.0264 | 0.0696 | 0.1192 | 0.1154 | 0.1472 | 0.5162 | 13 | 17 | 27 | 55 | 99 | 150 | 212 | 304 | 427 | 0.0207 | 22.64 | 5.797 | 0.4177 | 57133.8 | 26400000 | 14400000000 | 8750000000000 | 0.5240 | 0.1275 | 0.0365 | 0.0012 | 0.1204 | 0.0053 | 0.1762 | 0.0439 | 0.2018 | 0.1082 | 0.1883 | 0.1766 | 0.1249 | 0.1778 | 0.0762 | 0.1466 | 0.0532 | 0.1487 | 0.0224 | 0.1917 | 0.0006 | 0.0004 | 0.0018 | 0.0006 | 0.0042 | 0.0024 | 0.0165 | 0.0138 | 0.0564 | 0.0447 | 0.0762 | 0.0656 | 0.0665 | 0.0531 | 0.0911 | 0.0798 | 0.6869 | 0.7397 | 0.0013 | 0.0013 | 0.0019 | 0.0043 | 0.0055 | 0.0080 | 0.0249 | 0.0268 | 0.0675 | 0.0771 | 0.0949 | 0.1009 | 0.0777 | 0.0746 | 0.0971 | 0.0949 | 0.6292 | 0.6123 | 0.0004 | 0.0022 | 0.0050 | 0.0187 | 0.0604 | 0.0872 | 0.0731 | 0.1006 | 0.6523 |
| Hs 578T | Barasertib | 1.1 | uM | DRAQ5 | 1 | TMRE | 2 | 1 | 16 | 1 | 766 | 509 | | 21316 | 24107 | 152.8 | 47.18 | 163.56 | 211.64 | 92 | 112 | 127 | 140 | 153 | 165 | 177 | 192 | 213 | 0.1036 | 2498 | 0.827 | 32.25 | 8.06 | 7 | 0.0040 | 86 | 0.0005 | 77.74 | 7.966 | 0.1418 | 25560.0 | 4600000 | 879000000 | 178000000000 | 0.4877 | 0.1525 | 0.0009 | 0.0000 | 0.0037 | 0.0002 | 0.0149 | 0.0010 | 0.0428 | 0.0072 | 0.1047 | 0.0330 | 0.1809 | 0.0736 | 0.1588 | 0.0762 | 0.1780 | 0.0986 | 0.3152 | 0.7103 | 0.0003 | 0.0000 | 0.0008 | 0.0001 | 0.0020 | 0.0004 | 0.0097 | 0.0036 | 0.0325 | 0.0180 | 0.0642 | 0.0375 | 0.0588 | 0.0332 | 0.0797 | 0.0428 | 0.7519 | 0.8643 | 0.0029 | 0.0050 | 0.0051 | 0.0208 | 0.0156 | 0.0337 | 0.0478 | 0.0972 | 0.1088 | 0.1622 | 0.1603 | 0.2009 | 0.1202 | 0.1275 | 0.1473 | 0.1314 | 0.3919 | 0.2212 | 0.0008 | 0.0017 | 0.0048 | 0.0220 | 0.0553 | 0.0994 | 0.0941 | 0.1118 | 0.6100 | 16 | 20 | 29 | 40 | 58 | 89 | 164 | 305 | 506 | 0.0680 | 12.41 | 4.640 | 0.6115 | 71539.6 | 42800000 | 29400000000 | 22000000000000 | 0.5538 | 0.1336 | 0.0351 | 0.0046 | 0.1280 | 0.0167 | 0.2120 | 0.0578 | 0.1783 | 0.0940 | 0.1652 | 0.1624 | 0.1225 | 0.1970 | 0.0736 | 0.1265 | 0.0427 | 0.1262 | 0.0427 | 0.2147 | 0.0004 | 0.0008 | 0.0014 | 0.0014 | 0.0027 | 0.0031 | 0.0150 | 0.0104 | 0.0386 | 0.0411 | 0.0622 | 0.0561 | 0.0522 | 0.0433 | 0.0703 | 0.0687 | 0.7572 | 0.7752 | 0.0009 | 0.0010 | 0.0030 | 0.0044 | 0.0068 | 0.0054 | 0.0149 | 0.0123 | 0.0452 | 0.0465 | 0.0647 | 0.0707 | 0.0588 | 0.0625 | 0.0807 | 0.0936 | 0.7250 | 0.7037 | 0.0003 | 0.0026 | 0.0046 | 0.0144 | 0.0427 | 0.0684 | 0.0512 | 0.0708 | 0.7451 |
| MCF 10A | A443654 | 0.12 | uM | DRAQ5 | 1 | TMRE | 2 | 2 | 11 | 1 | 780 | 643 | | 4246 | 9503 | 153.2 | 43.23 | 163.95 | 111.35 | 107 | 118 | 127 | 135 | 144 | 155 | 167 | 184 | 213 | 0.0930 | 884 | 1.215 | 66.84 | 30.36 | 1 | 0.0445 | 189 | 0.0016 | 33.38 | 6.721 | 0.2068 | 25324.3 | 4540000 | 884000000 | 186000000000 | 0.4222 | 0.2177 | 0.0004 | 0.0000 | 0.0009 | 0.0000 | 0.0065 | 0.0005 | 0.0285 | 0.0037 | 0.1085 | 0.0264 | 0.1876 | 0.0650 | 0.1746 | 0.0647 | 0.2040 | 0.0836 | 0.2891 | 0.7561 | 0.0003 | 0.0000 | 0.0000 | 0.0000 | 0.0016 | 0.0002 | 0.0110 | 0.0012 | 0.0397 | 0.0171 | 0.0784 | 0.0293 | 0.0800 | 0.0238 | 0.1178 | 0.0358 | 0.6711 | 0.8927 | 0.0023 | 0.0000 | 0.0047 | 0.0049 | 0.0140 | 0.0196 | 0.0756 | 0.1225 | 0.1465 | 0.1716 | 0.1686 | 0.2059 | 0.1128 | 0.1152 | 0.1419 | 0.1127 | 0.3337 | 0.2475 | 0.0011 | 0.0022 | 0.0056 | 0.0332 | 0.0917 | 0.1507 | 0.1074 | 0.1277 | 0.4803 | 49 | 74 | 95 | 116 | 139 | 164 | 198 | 245 | 310 | 0.0019 | 44.15 | 6.783 | 0.2632 | 39278.6 | 12800000 | 5480000000 | 3000000000000 | 0.5562 | 0.1215 | 0.0241 | 0.0012 | 0.0805 | 0.0056 | 0.1411 | 0.0391 | 0.1416 | 0.0770 | 0.1754 | 0.1299 | 0.1546 | 0.1697 | 0.1157 | 0.1456 | 0.0995 | 0.1528 | 0.0676 | 0.2792 | 0.0014 | 0.0002 | 0.0026 | 0.0009 | 0.0069 | 0.0057 | 0.0242 | 0.0137 | 0.0746 | 0.0545 | 0.1063 | 0.0876 | 0.0950 | 0.0778 | 0.1295 | 0.1115 | 0.5595 | 0.6480 | 0.0031 | 0.0018 | 0.0045 | 0.0054 | 0.0118 | 0.0145 | 0.0478 | 0.0559 | 0.1069 | 0.1335 | 0.1491 | 0.1807 | 0.1301 | 0.1326 | 0.1557 | 0.1685 | 0.3910 | 0.3070 | 0.0018 | 0.0050 | 0.0089 | 0.0404 | 0.0908 | 0.1409 | 0.1049 | 0.1375 | 0.4699 |
| MCF 10A | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 266 | 832 | | 5052 | 10241 | 147.7 | 42.12 | 164.11 | 146.78 | 101 | 114 | 123 | 132 | 141 | 151 | 163 | 178 | 201 | 0.0842 | 862 | 1.052 | 93.96 | 28.02 | 1 | 0.0449 | 227 | 0.0015 | 34.75 | 6.782 | 0.2136 | 23601.0 | 4100000 | 775000000 | 160000000000 | 0.4351 | 0.2145 | 0.0000 | 0.0000 | 0.0014 | 0.0000 | 0.0119 | 0.0004 | 0.0418 | 0.0025 | 0.1162 | 0.0275 | 0.1757 | 0.0555 | 0.1934 | 0.0737 | 0.1916 | 0.1095 | 0.2680 | 0.7309 | 0.0000 | 0.0000 | 0.0005 | 0.0000 | 0.0016 | 0.0002 | 0.0152 | 0.0008 | 0.0452 | 0.0174 | 0.0714 | 0.0304 | 0.0903 | 0.0289 | 0.1092 | 0.0521 | 0.6665 | 0.8702 | 0.0029 | 0.0073 | 0.0164 | 0.0171 | 0.0299 | 0.0465 | 0.0598 | 0.1345 | 0.1583 | 0.1736 | 0.1631 | 0.1760 | 0.1361 | 0.1100 | 0.1544 | 0.1271 | 0.2790 | 0.2078 | 0.0023 | 0.0041 | 0.0120 | 0.0322 | 0.0989 | 0.1427 | 0.1141 | 0.1542 | 0.4395 | 13 | 30 | 59 | 89 | 123 | 168 | 218 | 280 | 374 | 0.0051 | 65.13 | 6.912 | 0.2905 | 48476.3 | 18800000 | 8740000000 | 4630000000000 | 0.4979 | 0.1489 | 0.0225 | 0.0023 | 0.1359 | 0.0100 | 0.2239 | 0.0492 | 0.1838 | 0.0904 | 0.1746 | 0.1755 | 0.1352 | 0.2178 | 0.0803 | 0.1586 | 0.0331 | 0.1509 | 0.0106 | 0.1453 | 0.0000 | 0.0002 | 0.0014 | 0.0012 | 0.0045 | 0.0043 | 0.0163 | 0.0104 | 0.0593 | 0.0502 | 0.0964 | 0.0849 | 0.0821 | 0.0672 | 0.1055 | 0.0971 | 0.6345 | 0.6846 | 0.0014 | 0.0028 | 0.0029 | 0.0077 | 0.0063 | 0.0120 | 0.0284 | 0.0359 | 0.0831 | 0.0921 | 0.1287 | 0.1354 | 0.1006 | 0.1051 | 0.1284 | 0.1343 | 0.5201 | 0.4747 | 0.0002 | 0.0029 | 0.0059 | 0.0176 | 0.0699 | 0.1148 | 0.0813 | 0.1176 | 0.5899 | ||
| SK-BR-3 | 0 | DRAQ5 | 1 | TMRE | 2 | 2 | 2 | 1 | 758 | 118 | | 3722 | 7678 | 368.8 | 182.51 | 164.24 | 272.94 | 145 | 178 | 217 | 266 | 351 | 446 | 510 | 563 | 614 | 0.0847 | 650 | 1.108 | 87.24 | 31.58 | 2 | 0.0623 | 232 | 0.0018 | 10.54 | 6.623 | 0.3115 | 169332.0 | 88000000 | 48900000000 | 28300000000000 | 0.2899 | 0.3386 | 0.0000 | 0.0007 | 0.0000 | 0.0027 | 0.0086 | 0.0047 | 0.0310 | 0.0167 | 0.1480 | 0.0670 | 0.2220 | 0.0965 | 0.1463 | 0.0810 | 0.1911 | 0.1186 | 0.2530 | 0.6122 | 0.0000 | 0.0000 | 0.0000 | 0.0008 | 0.0010 | 0.0020 | 0.0029 | 0.0035 | 0.0201 | 0.0203 | 0.0315 | 0.0250 | 0.0220 | 0.0238 | 0.0382 | 0.0355 | 0.8844 | 0.8892 | 0.0000 | 0.0009 | 0.0000 | 0.0009 | 0.0000 | 0.0019 | 0.0066 | 0.0149 | 0.0238 | 0.0411 | 0.0416 | 0.0747 | 0.0350 | 0.0691 | 0.0430 | 0.0756 | 0.8500 | 0.7208 | 0.0000 | 0.0000 | 0.0006 | 0.0017 | 0.0251 | 0.0345 | 0.0239 | 0.0395 | 0.8747 | 12 | 17 | 22 | 28 | 43 | 72 | 114 | 240 | 499 | 0.0621 | 27.12 | 4.594 | 0.6002 | 101458.0 | 93500000 | 101000000000 | 118000000000000 | 0.3873 | 0.2579 | 0.0278 | 0.0021 | 0.0732 | 0.0103 | 0.1995 | 0.0372 | 0.1692 | 0.0702 | 0.1843 | 0.1569 | 0.1162 | 0.1610 | 0.0909 | 0.1352 | 0.0707 | 0.1197 | 0.0682 | 0.3075 | 0.0019 | 0.0000 | 0.0014 | 0.0028 | 0.0053 | 0.0035 | 0.0101 | 0.0102 | 0.0483 | 0.0501 | 0.0718 | 0.0654 | 0.0565 | 0.0556 | 0.0775 | 0.0832 | 0.7271 | 0.7292 | 0.0000 | 0.0006 | 0.0041 | 0.0006 | 0.0053 | 0.0026 | 0.0077 | 0.0057 | 0.0543 | 0.0529 | 0.0721 | 0.0861 | 0.0543 | 0.0529 | 0.0874 | 0.0848 | 0.7147 | 0.7136 | 0.0005 | 0.0027 | 0.0086 | 0.0065 | 0.0507 | 0.0706 | 0.0507 | 0.0841 | 0.7256 |