BGJ398 KINOMEscan - Dataset (ID:20224)
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| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| BGJ398 | AAK1 | 76.0 | 1 | uM |
| BGJ398 | ABL1(E255K)-phosphorylated | 67.0 | 1 | uM |
| BGJ398 | ABL1(F317I)-nonphosphorylated | 87.0 | 1 | uM |
| BGJ398 | ABL1(F317I)-phosphorylated | 100.0 | 1 | uM |
| BGJ398 | ABL1(F317L)-nonphosphorylated | 73.0 | 1 | uM |
| BGJ398 | ABL1(F317L)-phosphorylated | 96.0 | 1 | uM |
| BGJ398 | ABL1(H396P)-nonphosphorylated | 19.0 | 1 | uM |
| BGJ398 | ABL1(H396P)-phosphorylated | 74.0 | 1 | uM |
| BGJ398 | ABL1(M351T)-phosphorylated | 81.0 | 1 | uM |
| BGJ398 | ABL1(Q252H)-nonphosphorylated | 28.0 | 1 | uM |
| BGJ398 | ABL1(Q252H)-phosphorylated | 80.0 | 1 | uM |
| BGJ398 | ABL1(T315I)-nonphosphorylated | 66.0 | 1 | uM |
| BGJ398 | ABL1(T315I)-phosphorylated | 92.0 | 1 | uM |
| BGJ398 | ABL1(Y253F)-phosphorylated | 72.0 | 1 | uM |
| BGJ398 | ABL1-nonphosphorylated | 55.0 | 1 | uM |
| BGJ398 | ABL1-phosphorylated | 64.0 | 1 | uM |
| BGJ398 | ABL2 | 62.0 | 1 | uM |
| BGJ398 | ACVR1 | 90.0 | 1 | uM |
| BGJ398 | ACVR1B | 89.0 | 1 | uM |
| BGJ398 | ACVR2A | 100.0 | 1 | uM |
| BGJ398 | ACVR2B | 100.0 | 1 | uM |
| BGJ398 | ACVRL1 | 74.0 | 1 | uM |
| BGJ398 | ADCK3 | 96.0 | 1 | uM |
| BGJ398 | ADCK4 | 99.0 | 1 | uM |
| BGJ398 | AKT1 | 98.0 | 1 | uM |