Ibrutinib KINOMEscan - Dataset (ID:20222)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Ibrutinib | ABL1(F317L)-phosphorylated | 48.0 | 1 | uM |
Ibrutinib | ABL1(F317L)-nonphosphorylated | 16.0 | 1 | uM |
Ibrutinib | ABL1(F317I)-phosphorylated | 39.0 | 1 | uM |
Ibrutinib | ABL1(F317I)-nonphosphorylated | 30.0 | 1 | uM |
Ibrutinib | ABL1(E255K)-phosphorylated | 65.0 | 1 | uM |
Ibrutinib | AAK1 | 92.0 | 1 | uM |