Ibrutinib KINOMEscan - Dataset (ID:20222)

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Small Molecule Protein % Control Assay compound conc Conc unit
Ibrutinib ABL1(F317L)-phosphorylated 48.0 1
uM
Ibrutinib ABL1(F317L)-nonphosphorylated 16.0 1
uM
Ibrutinib ABL1(F317I)-phosphorylated 39.0 1
uM
Ibrutinib ABL1(F317I)-nonphosphorylated 30.0 1
uM
Ibrutinib ABL1(E255K)-phosphorylated 65.0 1
uM
Ibrutinib AAK1 92.0 1
uM