Ibrutinib KINOMEscan - Dataset (ID:20222)

Proteins Studied

  • Page 1 of 19
  • 1 to 25 of 456 Proteins
LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200481 NEK10 200481 Q6ZWH5
NIMA (never in mitosis gene a)- related kinase 10
KINOMEscan
200470 BUB1 200470
Budding uninhibited by benzimidazoles 1 homolog (yeast); BUB1A; BUB1L; hBUB1
KINOMEscan
200476 SGK1 200476 O00141
Serine/threonine-protein kinase Sgk1; serum/glucocorticoid regulated kinase 1; SGK
KINOMEscan
201108 SGK2 201108 Q9HBY8
Serine/threonine-protein kinase Sgk2; Serum/glucocorticoid-regulated kinase 2
KINOMEscan
200477 WNK1 200477 Q9H4A3
WNK lysine deficient protein kinase 1; KDP; PSK; p65; HSN2; HSAN2; PRKWNK1
KINOMEscan
200471 CSF1R-autoinhibited 200471 P07333
Colony stimulating factor 1 receptor; CD115; C-FMS; CSF1R; CSF-1R; CSF-1-R; CSFR; FIM2; FIM-2; FMS; Fms/CSFR
KINOMEscan
200472 FLT3-autoinhibited 200472 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan
200475 RSK2(Kin.Dom.2-C-terminal) 200475 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KINOMEscan Kin.Dom.2-C-terminal
200479 ALK(C1156Y) 200479 Q9UM73
Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK
KINOMEscan C1156Y
201107 MAP3K14 201107 Q99558
Mitogen-activated protein kinase kinase kinase 14; NF-kappa-beta-inducing kinase; NIK
KINOMEscan
200480 ALK(L1196M) 200480 Q9UM73
Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK
KINOMEscan L1196M
200478 WNK3 200478 Q9BYP7
WNK lysine deficient protein kinase 3; PRKWNK3
KINOMEscan
200474 KIT-autoinhibited 200474 P10721
V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR
KINOMEscan
200473 HASP 200473 Q8TF76
Serine/threonine-protein kinase haspin; germ cell associated 2 (haspin); GSG2; HASPIN
KINOMEscan
200024 ABL1-nonphosphorylated 200024 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan nonphosphorylated Wild Type; Partial length
200038 AMPK-alpha1 200038 Q13131
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1
KINOMEscan Wild Type; Partial length
200045 AURKB 200045 Q96GD4
Aurora kinase B; AIK2; AIM1; AIM-1; ARK2; Aur1; AurB; AurB/Aur1; AURKB; aurkb-sv1; aurkb-sv2; IPL1; STK12; STK5
KINOMEscan Wild Type; Partial length
200040 ANKK1 200040 Q8NFD2
Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288
KINOMEscan Wild Type; Partial length
200044 AURKA 200044 O14965
Aurora kinase A; AIK; AIRK1; ARK1; Aur2; AURA; AurA/Aur2; AURKA; AURORA2; Aurora-A; Ayk1; BTAK; IAK; IAK1; MGC34538; STK15; STK6; STK7
KINOMEscan Wild Type; Partial length
200048 BIKE 200048 Q9NSY1
BMP2 inducible kinase; BIKE; BMP2K; DKFZp434K0614; DKFZp434P0116; HRIHFB2017
KINOMEscan Wild Type; Partial length
200049 BLK 200049 P51451
Tyrosine-protein kinase BLK; B lymphoid tyrosine kinase; BLK; MGC10442
KINOMEscan Wild Type; Partial length
200041 NUAK1 200041 O60285
NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1
KINOMEscan Wild Type; Partial length
200036 AKT3 200036 Q9Y243
V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2
KINOMEscan Wild Type; Partial length
200031 ACVRL1 200031 P37023
Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
KINOMEscan Wild Type; Partial length
200042 M3K5 200042 Q99683
Mitogen-activated protein kinase kinase kinase 5; ASK; ASK/MAP3K5; ASK1; MAP3K5; MAPKKK5; MEKK5
KINOMEscan Wild Type; Partial length
  • Page 1 of 19
  • 1 to 25 of 456 Proteins