Ibrutinib KINOMEscan - Dataset (ID:20222)
Proteins Studied
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LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200481 | NEK10 | 200481 | Q6ZWH5 | NIMA (never in mitosis gene a)- related kinase 10 | KINOMEscan | ||||
200470 | BUB1 | 200470 | Budding uninhibited by benzimidazoles 1 homolog (yeast); BUB1A; BUB1L; hBUB1 | KINOMEscan | |||||
200476 | SGK1 | 200476 | O00141 | Serine/threonine-protein kinase Sgk1; serum/glucocorticoid regulated kinase 1; SGK | KINOMEscan | ||||
201108 | SGK2 | 201108 | Q9HBY8 | Serine/threonine-protein kinase Sgk2; Serum/glucocorticoid-regulated kinase 2 | KINOMEscan | ||||
200477 | WNK1 | 200477 | Q9H4A3 | WNK lysine deficient protein kinase 1; KDP; PSK; p65; HSN2; HSAN2; PRKWNK1 | KINOMEscan | ||||
200471 | CSF1R-autoinhibited | 200471 | P07333 | Colony stimulating factor 1 receptor; CD115; C-FMS; CSF1R; CSF-1R; CSF-1-R; CSFR; FIM2; FIM-2; FMS; Fms/CSFR | KINOMEscan | ||||
200472 | FLT3-autoinhibited | 200472 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ||||
200475 | RSK2(Kin.Dom.2-C-terminal) | 200475 | P51812 | Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2 | KINOMEscan | Kin.Dom.2-C-terminal | |||
200479 | ALK(C1156Y) | 200479 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | C1156Y | |||
201107 | MAP3K14 | 201107 | Q99558 | Mitogen-activated protein kinase kinase kinase 14; NF-kappa-beta-inducing kinase; NIK | KINOMEscan | ||||
200480 | ALK(L1196M) | 200480 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | L1196M | |||
200478 | WNK3 | 200478 | Q9BYP7 | WNK lysine deficient protein kinase 3; PRKWNK3 | KINOMEscan | ||||
200474 | KIT-autoinhibited | 200474 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | ||||
200473 | HASP | 200473 | Q8TF76 | Serine/threonine-protein kinase haspin; germ cell associated 2 (haspin); GSG2; HASPIN | KINOMEscan | ||||
200024 | ABL1-nonphosphorylated | 200024 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | nonphosphorylated | Wild Type; Partial length | ||
200038 | AMPK-alpha1 | 200038 | Q13131 | Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1 | KINOMEscan | Wild Type; Partial length | |||
200045 | AURKB | 200045 | Q96GD4 | Aurora kinase B; AIK2; AIM1; AIM-1; ARK2; Aur1; AurB; AurB/Aur1; AURKB; aurkb-sv1; aurkb-sv2; IPL1; STK12; STK5 | KINOMEscan | Wild Type; Partial length | |||
200040 | ANKK1 | 200040 | Q8NFD2 | Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288 | KINOMEscan | Wild Type; Partial length | |||
200044 | AURKA | 200044 | O14965 | Aurora kinase A; AIK; AIRK1; ARK1; Aur2; AURA; AurA/Aur2; AURKA; AURORA2; Aurora-A; Ayk1; BTAK; IAK; IAK1; MGC34538; STK15; STK6; STK7 | KINOMEscan | Wild Type; Partial length | |||
200048 | BIKE | 200048 | Q9NSY1 | BMP2 inducible kinase; BIKE; BMP2K; DKFZp434K0614; DKFZp434P0116; HRIHFB2017 | KINOMEscan | Wild Type; Partial length | |||
200049 | BLK | 200049 | P51451 | Tyrosine-protein kinase BLK; B lymphoid tyrosine kinase; BLK; MGC10442 | KINOMEscan | Wild Type; Partial length | |||
200041 | NUAK1 | 200041 | O60285 | NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1 | KINOMEscan | Wild Type; Partial length | |||
200036 | AKT3 | 200036 | Q9Y243 | V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2 | KINOMEscan | Wild Type; Partial length | |||
200031 | ACVRL1 | 200031 | P37023 | Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I | KINOMEscan | Wild Type; Partial length | |||
200042 | M3K5 | 200042 | Q99683 | Mitogen-activated protein kinase kinase kinase 5; ASK; ASK/MAP3K5; ASK1; MAP3K5; MAPKKK5; MEKK5 | KINOMEscan | Wild Type; Partial length |