ZSTK474 KINOMEscan - Dataset (ID:20220)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200175 FLT4 200175 P35916
Fms-related tyrosine kinase 4; FLT4; FLT41; LMPH1A; PCL; VEGFR3
KINOMEscan Wild Type; Partial length
200458 VGFR2 200458 P35968
Vascular endothelial growth factor receptor 2; kinase insert domain receptor; CD309; FLK1; FLK-1; KDR; KRD-1; Ly73; VEGFR; VEGFR2; VEGFR-2
KINOMEscan Wild Type; Partial length
200252 MP2K2 200252 P36507
Dual specificity mitogen-activated protein kinase kinase 2; mitogen-activated protein kinase kinase 2; FLJ26075; MAP2K2; MAPKK2; MEK2; MEK2/MAP2K2; MKK2; PRKMK2
KINOMEscan Wild Type; Full length
200173 FLT3(N841I) 200173 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan N841I Mutation (N841I); Partial length
200171 FLT3(ITD) 200171 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan ITD Mutation (ITD); Partial length
200170 FLT3(D835Y) 200170 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan D835Y Mutation (D835Y); Partial length
200169 FLT3(D835H) 200169 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan D835H Mutation (D835H); Partial length
200168 FLT3 200168 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan Wild Type; Partial length
200172 FLT3(K663Q) 200172 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan K663Q Mutation (K663Q); Partial length
200050 BMPR1A 200050 P36894
Bone morphogenetic protein receptor, type IA; 10q23del; ACVRLK3; ALK3; BMPR1A; CD292; SKR5
KINOMEscan Wild Type; Partial length
200028 ACVR1B 200028 P36896
Activin A receptor, type IB; ACTRIB; ACVR1B; ACVRLK4; ALK4; SKR2
KINOMEscan Wild Type; Partial length
200433 TGFBR1 200433 P36897
Transforming growth factor, beta receptor 1; AAT5; ACVRLK4; ALK5; ALK-5; LDS1A; LDS2A; SKR4; TGFBR1; TGFR-1
KINOMEscan Wild Type; Partial length
200031 ACVRL1 200031 P37023
Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
KINOMEscan Wild Type; Partial length
200434 TGFBR2 200434 P37173
Transforming growth factor, beta receptor II (70/80kDa); AAT3; FAA3; LDS1B; LDS2B; MFS2; RIIC; TAAD2; TGFbeta-RII; TGFBR2; TGFR-2
KINOMEscan Wild Type; Partial length
200095 CSK 200095 P41240
C-src tyrosine kinase; CSK; MGC117393
KINOMEscan Wild Type; Full length
200323 PIK3CA 200323 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan Wild Type; Partial length
200327 PIK3CA(E545K) 200327 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E545K Mutation (E545K); Partial length
200333 PIK3CB 200333 P42338
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit beta; DKFZp779K1237; MGC133043; P110BETA; PI3K; PI3KBETA; PIK3C1; PIK3CB; PI3K-beta
KINOMEscan Wild Type; Partial length
200431 TEC 200431 P42680
Tyrosine-protein kinase Tec; MGC126760; MGC126762; PSCTK4; TEC
KINOMEscan Wild Type; Partial length
200449 TXK 200449 P42681
TXK tyrosine kinase; BTKL; MGC22473; PSCTK5; PTK4; RLK; TKL; TXK
KINOMEscan Wild Type; Partial length
200026 ABL2 200026 P42684
V-abl Abelson murine leukemia viral oncogene homolog 2 (arg, Abelson-related gene); ABL2; ABLL; ARG; FLJ22224; FLJ31718; FLJ41441
KINOMEscan Wild Type; Partial length
200176 FRK 200176 P42685
Tyrosine-protein kinase FRK; Fyn-related kinase; FRK; GTK; PTK5; RAK
KINOMEscan Wild Type; Partial length
200469 ZAP70 200469 P43403
Tyrosine-protein kinase ZAP-70; Zeta-chain (TCR) associated protein kinase 70kDa; FLJ17670; FLJ17679; SRK; STD; TZK; ZAP70; ZAP-70
KINOMEscan Wild Type; Partial length
200425 SYK 200425 P43405
Tyrosine-protein kinase SYK; spleen tyrosine kinase; p72-Syk; DKFZp313N1010; FLJ25043; FLJ37489; SYK
KINOMEscan Wild Type; Partial length
200211 JNK1 200211 P45983
Mitogen-activated protein kinase 8; JNK; JNK1; JNK1A2; JNK21B1/2; MAPK8; PRKM8; SAPK1
KINOMEscan Wild Type; Full length