DCC-2036 KiNativ -- single dose experiment - Dataset (ID:20210)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
DCC-2036 Ramos (RA 1) MAP3K1
DVKGANLLIDSTGQR
Lys2
88.6
 1
uM
DCC-2036 Ramos (RA 1) M3K2,MAP3K3
DIKGANILR
Lys2
-16.8
 1
uM
DCC-2036 Ramos (RA 1) MAP3K4
DIKGANIFLTSSGLIK
Lys2
4.2
 1
uM
DCC-2036 Ramos (RA 1) MAP3K5
DIKGDNVLINTYSGVLK
Lys2
9.8
 1
uM
DCC-2036 Ramos (RA 1) MARK2,MARK3
DLKAENLLLDADMNIK
Lys2
6.2
 1
uM
DCC-2036 Ramos (RA 1) MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
-11.1
 1
uM
DCC-2036 Ramos (RA 1) MAST3
DLKPDNLLITSLGHIK
Lys2
26.2
 1
uM
DCC-2036 Ramos (RA 1) MASTL
LYAVKVVK
Lys1
-2.9
 1
uM
DCC-2036 Ramos (RA 1) MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
-2.1
 1
uM
DCC-2036 Ramos (RA 1) MST2
ESGQVVAIKQVPVESDLQEIIK
Lys1
0.9
 1
uM
DCC-2036 Ramos (RA 1) MST3
DIKAANVLLSEHGEVK
Lys2
8.1
 1
uM
DCC-2036 Ramos (RA 1) MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
19.0
 1
uM
DCC-2036 Ramos (RA 1) NDR1
DTGHVYAMKILR
Lys1
-12.4
 1
uM
DCC-2036 Ramos (RA 1) NDR2
DIKPDNLLLDAK
Lys2
-7.5
 1
uM
DCC-2036 Ramos (RA 1) NEK3
SKNIFLTQNGK
Activation Loop
4.6
 1
uM
DCC-2036 Ramos (RA 1) NEK6,NEK7
DIKPANVFITATGVVK
Lys2
13.0
 1
uM
DCC-2036 Ramos (RA 1) NEK7
AACLLDGVPVALKK
Lys1
1.6
 1
uM
DCC-2036 Ramos (RA 1) NEK9
DIKTLNIFLTK
Lys2
0.5
 1
uM
DCC-2036 Ramos (RA 1) MK14
QELNKTIWEVPER
Protein Kinase Domain
69.6
 1
uM
DCC-2036 Ramos (RA 1) p38d,p38g
DLKPGNLAVNEDCELK
Lys2
57.6
 1
uM
DCC-2036 Ramos (RA 1) KS6B1
DLKPENIMLNHQGHVK
Lys2
-16.9
 1
uM
DCC-2036 Ramos (RA 1) CDK14
LVALKVIR
Lys1
94.2
 1
uM
DCC-2036 Ramos (RA 1) PI4KB
VPHTQAVVLNSKDK
ATP
-10.6
 1
uM
DCC-2036 Ramos (RA 1) PIK3C3
TEDGGKYPVIFKHGDDLR
ATP
-6.5
 1
uM
DCC-2036 Ramos (RA 1) PIK3CB
VFGEDSVGVIFKNGDDLR
ATP
1.2
 1
uM