QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 MWCL.1 SMG1
DTVTIHSVGGTITILPTKTKPK
ATP
2.026402071
1
uM
QL-XII-47 MWCL.1 SNRK
DLKPENVVFFEK
Lys2
17.0299839
1
uM
QL-XII-47 MWCL.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
-16.87895726
1
uM
QL-XII-47 MWCL.1 SRPK1/2
FVAMKVVK
Lys1
-11.61360647
1
uM
QL-XII-47 MWCL.1 STLK5
YSVKVLPWLSPEVLQQNLQGYDAK
Activation Loop
-1.488167509
1
uM
QL-XII-47 MWCL.1 STLK6
HTPTGTLVTIKITNLENCNEER
Lys1
-27.19332598
1
uM
QL-XII-47 MWCL.1 SYK
ISDFGLSKALR
Activation Loop
9.937407948
1
uM
QL-XII-47 MWCL.1 MAP3K7,TAK1
DLKPPNLLLVAGGTVLK
Lys2
4.848341421
1
uM
QL-XII-47 MWCL.1 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
-11.09760984
1
uM
QL-XII-47 MWCL.1 TAOK2
DVKAGNILLSEPGLVK
Lys2
-17.69969794
1
uM
QL-XII-47 MWCL.1 TBK1
TGDLFAIKVFNNISFLRPVDVQMR
Lys1
0.073270679
1
uM
QL-XII-47 MWCL.1 TEC
YVLDDQYTSSSGAKFPVK
Activation Loop
60.11680682
1
uM
QL-XII-47 MWCL.1 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
Lys2
-1.435121129
1
uM
QL-XII-47 MWCL.1 TLK1/2
YLNEIKPPIIHYDLKPGNILLVNGTACGEIK
Lys2
-2.951577221
1
uM
QL-XII-47 MWCL.1 ULK1
DLKPQNILLSNPAGR
Lys2
-14.58312377
1
uM
QL-XII-47 MWCL.1 ULK3
NISHLDLKPQNILLSSLEKPHLK
Lys2
2.928063615
1
uM
QL-XII-47 MWCL.1 VRK2
MLDVLEYIHENEYVHGDIKAANLLLGYK
Lys2
22.7412435
1
uM
QL-XII-47 MWCL.1 WEE1
YIHSMSLVHMDIKPSNIFISR
Lys2
-37.77693454
1
uM
QL-XII-47 MWCL.1 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
Lys2
-10.55702775
1
uM
QL-XII-47 MWCL.1 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
Lys2
-26.32668943
1
uM
QL-XII-47 MWCL.1 ZC2/TNIK
TGQLAAIKVMDVTGDEEEEIKQEINMLKK
Lys1
-2.724092946
1
uM
QL-XII-47 BCWM.1 ABL,ARG
LMTGDTYTAHAGAKFPIK
Activation Loop
-4.884271122
1
uM
QL-XII-47 BCWM.1 ABL,ARG
YSLTVAVKTLKEDTMEVEEFLK
Lys1
23.94636209
1
uM
QL-XII-47 BCWM.1 ACK
TVSVAVKCLKPDVLSQPEAMDDFIR
Lys1
16.75144083
1
uM
QL-XII-47 BCWM.1 AMPKa1,AMPKa2
DLKPENVLLDAHMNAK
Lys2
18.43323382
1
uM