QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | MWCL.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 2.026402071 | 1 | uM |
QL-XII-47 | MWCL.1 | SNRK | DLKPENVVFFEK | Lys2 | 17.0299839 | 1 | uM |
QL-XII-47 | MWCL.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -16.87895726 | 1 | uM |
QL-XII-47 | MWCL.1 | SRPK1/2 | FVAMKVVK | Lys1 | -11.61360647 | 1 | uM |
QL-XII-47 | MWCL.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | -1.488167509 | 1 | uM |
QL-XII-47 | MWCL.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | -27.19332598 | 1 | uM |
QL-XII-47 | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 9.937407948 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | 4.848341421 | 1 | uM |
QL-XII-47 | MWCL.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | -11.09760984 | 1 | uM |
QL-XII-47 | MWCL.1 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | -17.69969794 | 1 | uM |
QL-XII-47 | MWCL.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 0.073270679 | 1 | uM |
QL-XII-47 | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 60.11680682 | 1 | uM |
QL-XII-47 | MWCL.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -1.435121129 | 1 | uM |
QL-XII-47 | MWCL.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -2.951577221 | 1 | uM |
QL-XII-47 | MWCL.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -14.58312377 | 1 | uM |
QL-XII-47 | MWCL.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 2.928063615 | 1 | uM |
QL-XII-47 | MWCL.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 22.7412435 | 1 | uM |
QL-XII-47 | MWCL.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | -37.77693454 | 1 | uM |
QL-XII-47 | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.55702775 | 1 | uM |
QL-XII-47 | MWCL.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | -26.32668943 | 1 | uM |
QL-XII-47 | MWCL.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | -2.724092946 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 23.94636209 | 1 | uM |
QL-XII-47 | BCWM.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 16.75144083 | 1 | uM |
QL-XII-47 | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 18.43323382 | 1 | uM |