QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | MWCL.1 | FRK | HEIKLPVK | Activation Loop | 7.187023655 | 1 | uM |
| QL-XII-47 | BCWM.1 | FRK | HEIKLPVK | Activation Loop | -7.289586984 | 1 | uM |
| QL-XII-47 | BCWM.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | -27.19332598 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -87.4730226 | 1 | uM |
| QL-XII-47 | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -55.6912494 | 1 | uM |
| QL-XII-47 | MWCL.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -20.94285661 | 1 | uM |
| QL-XII-47 | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | ND | 1 | uM |
| QL-XII-47 | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 0.574708889 | 1 | uM |
| QL-XII-47 | MWCL.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | -4.184361 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -9.341503001 | 1 | uM |
| QL-XII-47 | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -18.81736377 | 1 | uM |
| QL-XII-47 | MWCL.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | ND | 1 | uM |
| QL-XII-47 | BCWM.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | 47.0732956 | 1 | uM |
| QL-XII-47 | MWCL.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -16.87895726 | 1 | uM |
| QL-XII-47 | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 0.388055572 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | -10.45585154 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | 8.135028611 | 1 | uM |
| QL-XII-47 | MWCL.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | -6.530594283 | 1 | uM |
| QL-XII-47 | BCWM.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 0.853020424 | 1 | uM |
| QL-XII-47 | MWCL.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 3.265960592 | 1 | uM |
| QL-XII-47 | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -4.698942545 | 1 | uM |
| QL-XII-47 | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 9.937407948 | 1 | uM |
| QL-XII-47 | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | 7.40661852 | 1 | uM |
| QL-XII-47 | BCWM.1 | DNAPK | KGGSWIQEINVAEK | ATP | -13.80369189 | 1 | uM |