QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 CaMK2g
TSTQEYAAKIINTK
Lys1
4.50076179
1
uM
QL-XII-47 MWCL.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
4.501665604
1
uM
QL-XII-47 BCWM.1 ARAF
DLKSNNIFLHEGLTVK
Lys2
4.534711447
1
uM
QL-XII-47 MWCL.1 PIK3CD
VNWLAHNVSKDNRQ
ATP
4.546978964
1
uM
QL-XII-47 MWCL.1 MP2K7
DVKPSNILLDER
Lys2
-45.5174114
1
uM
QL-XII-47 BCWM.1 LATS1
ALYATKTLR
Lys1
4.639137919
1
uM
QL-XII-47 BCWM.1 RSKL1_domain1
VLGVIDKVLLVMDTR
ATP
46.48841594
1
uM
QL-XII-47 MWCL.1 ABL,ARG
LMTGDTYTAHAGAKFPIK
Activation Loop
-4.6555368
1
uM
QL-XII-47 BCWM.1 MSK2 domain1
DLKLENVLLDSEGHIVLTDFGLSK
Lys2
-46.59383779
1
uM
QL-XII-47 MWCL.1 MAP2K4
DIKPSNILLDR
Lys2
-4.661208852
1
uM
QL-XII-47 BCWM.1 FRAP1
IQSIAPSLQVITSKQRPR
ATP
-4.698942545
1
uM
QL-XII-47 BCWM.1 BLK
IIDSEYTAQEGAKFPIK
Activation Loop
47.0732956
1
uM
QL-XII-47 BCWM.1 MST4
TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK
Lys1
4.712110007
1
uM
QL-XII-47 BCWM.1 MAP3K1
DVKGANLLIDSTGQR
Lys2
-4.774099061
1
uM
QL-XII-47 MWCL.1 RSK2 domain1
DLKPENILLDEEGHIKLTDFGLSKESIDHEK
Lys2
-48.46241013
1
uM
QL-XII-47 MWCL.1 MAP3K7,TAK1
DLKPPNLLLVAGGTVLK
Lys2
4.848341421
1
uM
QL-XII-47 BCWM.1 ABL,ARG
LMTGDTYTAHAGAKFPIK
Activation Loop
-4.884271122
1
uM
QL-XII-47 BCWM.1 MAP3K5
DIKGDNVLINTYSGVLK
Lys2
-4.886038638
1
uM
QL-XII-47 BCWM.1 ITPK1
ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR
ATP
49.00978471
1
uM
QL-XII-47 MWCL.1 MASTL
LYAVKVVK
Lys1
-4.9183009
1
uM
QL-XII-47 BCWM.1 PIK3CG
KKPLWLEFK
ATP
-49.28259781
1
uM
QL-XII-47 MWCL.1 GCN2_domain2
DLKPVNIFLDSDDHVK
Lys2
-49.83844146
1
uM
QL-XII-47 BCWM.1 MAST1,MAST2
DLKPDNLLITSMGHIK
Lys2
-49.97672913
1
uM
QL-XII-47 MWCL.1 RIPK2
VQVAVKHLHIHTPLLDSER
Lys1
5.017497496
1
uM
QL-XII-47 MWCL.1 KC1A
DIKPDNFLMGIGR
Lys2
-5.104906235
1
uM