QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -59.65168038 | 1 | uM |
QL-XII-47 | BCWM.1 | GCK | DIKGANLLLTLQGDVK | Lys2 | -3.557207356 | 1 | uM |
QL-XII-47 | BCWM.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | -73.95597608 | 1 | uM |
QL-XII-47 | BCWM.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | -12.56740412 | 1 | uM |
QL-XII-47 | BCWM.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | 2.952147748 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 23.94636209 | 1 | uM |
QL-XII-47 | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 18.43323382 | 1 | uM |
QL-XII-47 | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 4.534711447 | 1 | uM |
QL-XII-47 | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | 7.861261294 | 1 | uM |
QL-XII-47 | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -22.46332421 | 1 | uM |
QL-XII-47 | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 70.55327861 | 1 | uM |
QL-XII-47 | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 0.033712822 | 1 | uM |
QL-XII-47 | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -11.32754424 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 14.74034939 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -9.229049081 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 4.004453656 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | 11.68818243 | 1 | uM |
QL-XII-47 | BCWM.1 | CHK1 | DIKPENLLLDER | Lys2 | 2.996204004 | 1 | uM |
QL-XII-47 | BCWM.1 | KC1A | DIKPDNFLMGIGR | Lys2 | 5.412904442 | 1 | uM |
QL-XII-47 | BCWM.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | 16.73486558 | 1 | uM |
QL-XII-47 | BCWM.1 | eEF2K | YIKYNSNSGFVR | ATP | 21.43479928 | 1 | uM |
QL-XII-47 | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | -24.56149352 | 1 | uM |
QL-XII-47 | BCWM.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 39.74033143 | 1 | uM |
QL-XII-47 | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | 1.096021819 | 1 | uM |