QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 FGR
LIKDDEYNPCQGSKFPIK
Activation Loop
-59.65168038
1
uM
QL-XII-47 BCWM.1 GCK
DIKGANLLLTLQGDVK
Lys2
-3.557207356
1
uM
QL-XII-47 BCWM.1 GCN2_domain2
DLKPVNIFLDSDDHVK
Lys2
-73.95597608
1
uM
QL-XII-47 BCWM.1 GSK3B
DIKPQNLLLDPDTAVLK
Lys2
-12.56740412
1
uM
QL-XII-47 BCWM.1 HPK1
DIKGANILINDAGEVR
Lys2
2.952147748
1
uM
QL-XII-47 BCWM.1 ABL,ARG
LMTGDTYTAHAGAKFPIK
Activation Loop
-4.884271122
1
uM
QL-XII-47 BCWM.1 ABL,ARG
YSLTVAVKTLKEDTMEVEEFLK
Lys1
23.94636209
1
uM
QL-XII-47 BCWM.1 AMPKa1,AMPKa2
DLKPENVLLDAHMNAK
Lys2
18.43323382
1
uM
QL-XII-47 BCWM.1 ARAF
DLKSNNIFLHEGLTVK
Lys2
4.534711447
1
uM
QL-XII-47 BCWM.1 AurB
SHFIVALKVLFK
Lys1
7.861261294
1
uM
QL-XII-47 BCWM.1 BARK1
DLKPANILLDEHGHVR
Lys2
-22.46332421
1
uM
QL-XII-47 BCWM.1 BTK
YVLDDEYTSSVGSKFPVR
Activation Loop
70.55327861
1
uM
QL-XII-47 BCWM.1 CAMK1D
LFAVKCIPK
Lys1
0.033712822
1
uM
QL-XII-47 BCWM.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-11.32754424
1
uM
QL-XII-47 BCWM.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
14.74034939
1
uM
QL-XII-47 BCWM.1 CDK4
DLKPENILVTSGGTVK
Lys2
-9.229049081
1
uM
QL-XII-47 BCWM.1 CDK5
DLKPQNLLINR
Lys2
4.004453656
1
uM
QL-XII-47 BCWM.1 CDK9
DMKAANVLITR
Lys2
11.68818243
1
uM
QL-XII-47 BCWM.1 CHK1
DIKPENLLLDER
Lys2
2.996204004
1
uM
QL-XII-47 BCWM.1 KC1A
DIKPDNFLMGIGR
Lys2
5.412904442
1
uM
QL-XII-47 BCWM.1 CK2a2
DVKPHNVMIDHQQK
Lys2
16.73486558
1
uM
QL-XII-47 BCWM.1 eEF2K
YIKYNSNSGFVR
ATP
21.43479928
1
uM
QL-XII-47 BCWM.1 EPHB2
FLEDDTSDPTYTSALGGKIPIR
Activation Loop
-24.56149352
1
uM
QL-XII-47 BCWM.1 IRAK1
AIQFLHQDSPSLIHGDIKSSNVLLDER
Lys2
39.74033143
1
uM
QL-XII-47 BCWM.1 ILK
WQGNDIVVKVLK
Lys1
1.096021819
1
uM