QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 MWCL.1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
-17.67799308
1
uM
QL-XII-47 MWCL.1 PI42C
TLVIKEVSSEDIADMHSNLSNYHQYIVK
ATP
2.368941706
1
uM
QL-XII-47 MWCL.1 FYV1
GGKSGAAFYATEDDRFILK
ATP
11.54045713
1
uM
QL-XII-47 MWCL.1 PITSLRE
DLKTSNLLLSHAGILK
Lys2
-29.23162594
1
uM
QL-XII-47 MWCL.1 PKD2
DVAVKVIDK
Lys1
1.687843861
1
uM
QL-XII-47 MWCL.1 PKD3
DVAIKVIDK
Lys1
16.99061532
1
uM
QL-XII-47 MWCL.1 PKN1
VLLSEFRPSGELFAIKALK
Lys1
22.89169441
1
uM
QL-XII-47 MWCL.1 PKR
DLKPSNIFLVDTK
Lys2
-5.625731683
1
uM
QL-XII-47 MWCL.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
8.755945296
1
uM
QL-XII-47 MWCL.1 PRP4
CNILHADIKPDNILVNESK
Lys2
-61.44506492
1
uM
QL-XII-47 MWCL.1 PRPK
FLSGLELVKQGAEAR
ATP Loop
-21.99502308
1
uM
QL-XII-47 MWCL.1 FAK2
YIEDEDYYKASVTR
Activation Loop
-31.93905936
1
uM
QL-XII-47 MWCL.1 RAF1
DMKSNNIFLHEGLTVK
Lys2
7.81337788
1
uM
QL-XII-47 MWCL.1 RIPK2
VQVAVKHLHIHTPLLDSER
Lys1
5.017497496
1
uM
QL-XII-47 MWCL.1 RIPK3
DLKPSNVLLDPELHVK
Lys2
-13.02157961
1
uM
QL-XII-47 MWCL.1 ROCK1,ROCK2
DVKPDNMLLDK
Lys2
-14.23267034
1
uM
QL-XII-47 MWCL.1 RSK1 domain1
DLKPENILLDEEGHIKLTDFGLSKEAIDHEK
Lys2
-44.09153868
1
uM
QL-XII-47 MWCL.1 RSK1_domain2
DLKPSNILYVDESGNPECLR
Lys2
5.411076459
1
uM
QL-XII-47 MWCL.1 RSK1,RSK2,RSK3_domain1
DLKPENILLDEEGHIK
Lys2
-24.39230683
1
uM
QL-XII-47 MWCL.1 RSK2_domain2
DLKPSNILYVDESGNPESIR
Lys2
7.226741044
1
uM
QL-XII-47 MWCL.1 RSK3_domain1
DLKPENILLDEEGHIKITDFGLSK
Lys2
-22.55817594
1
uM
QL-XII-47 MWCL.1 RSK4 domain1
DLKPENILLDEIGHIK
Lys2
ND
1
uM
QL-XII-47 MWCL.1 RSKL1_domain1
VLGVIDKVLLVMDTR
ATP
22.96800436
1
uM
QL-XII-47 MWCL.1 SGK3
FYAVKVLQK
Lys1
9.129996049
1
uM
QL-XII-47 MWCL.1 SLK
DLKAGNILFTLDGDIK
Lys2
1.020533171
1
uM