QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | MWCL.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -17.67799308 | 1 | uM |
QL-XII-47 | MWCL.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | 2.368941706 | 1 | uM |
QL-XII-47 | MWCL.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 11.54045713 | 1 | uM |
QL-XII-47 | MWCL.1 | PITSLRE | DLKTSNLLLSHAGILK | Lys2 | -29.23162594 | 1 | uM |
QL-XII-47 | MWCL.1 | PKD2 | DVAVKVIDK | Lys1 | 1.687843861 | 1 | uM |
QL-XII-47 | MWCL.1 | PKD3 | DVAIKVIDK | Lys1 | 16.99061532 | 1 | uM |
QL-XII-47 | MWCL.1 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | 22.89169441 | 1 | uM |
QL-XII-47 | MWCL.1 | PKR | DLKPSNIFLVDTK | Lys2 | -5.625731683 | 1 | uM |
QL-XII-47 | MWCL.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 8.755945296 | 1 | uM |
QL-XII-47 | MWCL.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | -61.44506492 | 1 | uM |
QL-XII-47 | MWCL.1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | -21.99502308 | 1 | uM |
QL-XII-47 | MWCL.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -31.93905936 | 1 | uM |
QL-XII-47 | MWCL.1 | RAF1 | DMKSNNIFLHEGLTVK | Lys2 | 7.81337788 | 1 | uM |
QL-XII-47 | MWCL.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 5.017497496 | 1 | uM |
QL-XII-47 | MWCL.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -13.02157961 | 1 | uM |
QL-XII-47 | MWCL.1 | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | -14.23267034 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | -44.09153868 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK1_domain2 | DLKPSNILYVDESGNPECLR | Lys2 | 5.411076459 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | -24.39230683 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | 7.226741044 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK3_domain1 | DLKPENILLDEEGHIKITDFGLSK | Lys2 | -22.55817594 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | ND | 1 | uM |
QL-XII-47 | MWCL.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | 22.96800436 | 1 | uM |
QL-XII-47 | MWCL.1 | SGK3 | FYAVKVLQK | Lys1 | 9.129996049 | 1 | uM |
QL-XII-47 | MWCL.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 1.020533171 | 1 | uM |