CGP74514A KINOMEscan - Dataset (ID:20203)

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Small Molecule Protein % Control Assay compound conc Conc unit
CGP74514A ABL1(F317L)-phosphorylated 5.6 10
uM
CGP74514A ABL1(F317L)-nonphosphorylated 23.0 10
uM
CGP74514A ABL1(F317I)-phosphorylated 14.0 10
uM
CGP74514A ABL1(F317I)-nonphosphorylated 35.0 10
uM
CGP74514A ABL1(E255K)-phosphorylated 2.5 10
uM
CGP74514A AAK1 98.0 10
uM