CGP74514A KINOMEscan - Dataset (ID:20203)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| CGP74514A | AMPK-alpha1 | 22.0 | 10 | uM |
| CGP74514A | ALK(L1196M) | 28.0 | 10 | uM |
| CGP74514A | ALK(C1156Y) | 17.0 | 10 | uM |
| CGP74514A | ALK | 7.9 | 10 | uM |
| CGP74514A | AKT3 | 100.0 | 10 | uM |
| CGP74514A | AKT2 | 90.0 | 10 | uM |
| CGP74514A | AKT1 | 99.0 | 10 | uM |
| CGP74514A | ADCK4 | 71.0 | 10 | uM |
| CGP74514A | ADCK3 | 100.0 | 10 | uM |
| CGP74514A | ACVRL1 | 100.0 | 10 | uM |
| CGP74514A | ACVR2B | 100.0 | 10 | uM |
| CGP74514A | ACVR2A | 97.0 | 10 | uM |
| CGP74514A | ACVR1B | 100.0 | 10 | uM |
| CGP74514A | ACVR1 | 100.0 | 10 | uM |
| CGP74514A | ABL2 | 21.0 | 10 | uM |
| CGP74514A | ABL1(Y253F)-phosphorylated | 1.6 | 10 | uM |
| CGP74514A | ABL1(T315I)-phosphorylated | 17.0 | 10 | uM |
| CGP74514A | ABL1(T315I)-nonphosphorylated | 41.0 | 10 | uM |
| CGP74514A | ABL1(Q252H)-phosphorylated | 1.4 | 10 | uM |
| CGP74514A | ABL1(Q252H)-nonphosphorylated | 0.4 | 10 | uM |
| CGP74514A | ABL1-phosphorylated | 3.4 | 10 | uM |
| CGP74514A | ABL1-nonphosphorylated | 7.4 | 10 | uM |
| CGP74514A | ABL1(M351T)-phosphorylated | 3.8 | 10 | uM |
| CGP74514A | ABL1(H396P)-phosphorylated | 1.8 | 10 | uM |
| CGP74514A | ABL1(H396P)-nonphosphorylated | 0.1 | 10 | uM |