Imatinib KINOMEscan - Dataset (ID:20198)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Imatinib | BLK | 520.0 | nM |
Imatinib | KIT(D816H) | 560.0 | nM |
Imatinib | ABL1(F317I)-phosphorylated | 580.0 | nM |
Imatinib | LYN | 890.0 | nM |
Imatinib | HIPK4 | 960.0 | nM |
Imatinib | KIT(D816V) | 980.0 | nM |
Imatinib | GAK | 1000.0 | nM |
Imatinib | IRAK1 | 1200.0 | nM |
Imatinib | EPHA8 | 1400.0 | nM |
Imatinib | FRK | 1500.0 | nM |
Imatinib | RAF1 | 1700.0 | nM |
Imatinib | MELK | 1900.0 | nM |
Imatinib | CLK4 | 2100.0 | nM |
Imatinib | FGR | 2400.0 | nM |
Imatinib | KIT(V559D,T670I) | 2500.0 | nM |
Imatinib | MLTK | 2600.0 | nM |
Imatinib | JNK3 | 3100.0 | nM |
Imatinib | FYN | 3100.0 | nM |
Imatinib | BRAF(V600E) | 3300.0 | nM |
Imatinib | TNNI3K | 4300.0 | nM |
Imatinib | CLK1 | 4500.0 | nM |
Imatinib | JNK1 | 5000.0 | nM |
Imatinib | DRAK1 | 5300.0 | nM |
Imatinib | CDK11 | 5500.0 | nM |
Imatinib | FLT3(ITD) | 6300.0 | nM |