Imatinib KINOMEscan - Dataset (ID:20198)

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Small Molecule Protein Kd Conc unit
Imatinib BLK 520.0
nM
Imatinib KIT(D816H) 560.0
nM
Imatinib ABL1(F317I)-phosphorylated 580.0
nM
Imatinib LYN 890.0
nM
Imatinib HIPK4 960.0
nM
Imatinib KIT(D816V) 980.0
nM
Imatinib GAK 1000.0
nM
Imatinib IRAK1 1200.0
nM
Imatinib EPHA8 1400.0
nM
Imatinib FRK 1500.0
nM
Imatinib RAF1 1700.0
nM
Imatinib MELK 1900.0
nM
Imatinib CLK4 2100.0
nM
Imatinib FGR 2400.0
nM
Imatinib KIT(V559D,T670I) 2500.0
nM
Imatinib MLTK 2600.0
nM
Imatinib JNK3 3100.0
nM
Imatinib FYN 3100.0
nM
Imatinib BRAF(V600E) 3300.0
nM
Imatinib TNNI3K 4300.0
nM
Imatinib CLK1 4500.0
nM
Imatinib JNK1 5000.0
nM
Imatinib DRAK1 5300.0
nM
Imatinib CDK11 5500.0
nM
Imatinib FLT3(ITD) 6300.0
nM