Imatinib KINOMEscan - Dataset (ID:20198)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Imatinib | FES | nM | |
Imatinib | FGFR1 | nM | |
Imatinib | FGFR2 | nM | |
Imatinib | FGFR3 | nM | |
Imatinib | FGFR3(G697C) | nM | |
Imatinib | FGFR4 | nM | |
Imatinib | FGR | 2400.0 | nM |
Imatinib | VGFR1 | nM | |
Imatinib | FLT3 | nM | |
Imatinib | FLT3(D835H) | nM | |
Imatinib | FLT3(D835Y) | nM | |
Imatinib | FLT3(ITD) | 6300.0 | nM |
Imatinib | FLT3(K663Q) | nM | |
Imatinib | FLT3(N841I) | nM | |
Imatinib | FLT3(R834Q) | nM | |
Imatinib | FLT4 | nM | |
Imatinib | FRK | 1500.0 | nM |
Imatinib | FYN | 3100.0 | nM |
Imatinib | GAK | 1000.0 | nM |
Imatinib | GCN2(Kin.Dom.2,S808G) | nM | |
Imatinib | GRK1 | nM | |
Imatinib | GRK4 | nM | |
Imatinib | GRK7 | nM | |
Imatinib | GSK3A | nM | |
Imatinib | GSK3B | nM |