Dasatinib KINOMEscan - Dataset (ID:20196)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Dasatinib | ABL1(F317L)-phosphorylated | 0.02 | nM |
Dasatinib | ABL1(M351T)-phosphorylated | 0.02 | nM |
Dasatinib | ABL1(F317L)-nonphosphorylated | 0.03 | nM |
Dasatinib | ABL1(H396P)-nonphosphorylated | 0.03 | nM |
Dasatinib | ABL1-nonphosphorylated | 0.03 | nM |
Dasatinib | ABL1(Q252H)-nonphosphorylated | 0.04 | nM |
Dasatinib | ABL1(F317I)-phosphorylated | 0.04 | nM |
Dasatinib | EPHB6 | 0.04 | nM |
Dasatinib | ABL1(E255K)-phosphorylated | 0.05 | nM |
Dasatinib | ABL1-phosphorylated | 0.05 | nM |
Dasatinib | ABL1(H396P)-phosphorylated | 0.05 | nM |
Dasatinib | ABL1(Y253F)-phosphorylated | 0.06 | nM |
Dasatinib | ABL1(Q252H)-phosphorylated | 0.06 | nM |
Dasatinib | EPHA3 | 0.09 | nM |
Dasatinib | ABL1(F317I)-nonphosphorylated | 0.10 | nM |
Dasatinib | ABL2 | 0.17 | nM |
Dasatinib | LCK | 0.20 | nM |
Dasatinib | SRC | 0.21 | nM |
Dasatinib | BLK | 0.21 | nM |
Dasatinib | EPHA5 | 0.24 | nM |
Dasatinib | EPHA8 | 0.24 | nM |
Dasatinib | YES | 0.30 | nM |
Dasatinib | FRK | 0.31 | nM |
Dasatinib | EPHB4 | 0.34 | nM |
Dasatinib | HCK | 0.35 | nM |