AT-7519 KINOMEscan - Dataset (ID:20191)

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Small Molecule Protein Kd Conc unit
AT-7519 CASK 24.0
nM
AT-7519 GSK3A 23.0
nM
AT-7519 CDK4-cyclinD1 20.0
nM
AT-7519 CDK14 16.0
nM
AT-7519 PCTK3 14.0
nM
AT-7519 CDK4-cyclinD3 12.0
nM
AT-7519 GSK3B 11.0
nM
AT-7519 CDC2L1 8.4
nM
AT-7519 ICK 8.3
nM
AT-7519 CDK9 5.8
nM
AT-7519 CDC2L2 5.2
nM
AT-7519 CDC2L5 3.2
nM
AT-7519 CDK7 2.8
nM
AT-7519 CDKL5 2.6
nM
AT-7519 CDK16 1.1
nM
AT-7519 PCTK2 1.0
nM
AT-7519 ANKK1
nM
AT-7519 AMPK-alpha2
nM
AT-7519 ABL1-nonphosphorylated
nM
AT-7519 AMPK-alpha1
nM
AT-7519 ALK
nM
AT-7519 ABL1(Y253F)-phosphorylated
nM
AT-7519 ABL1(H396P)-nonphosphorylated
nM
AT-7519 AKT3
nM
AT-7519 AKT2
nM