CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | TAK1 | 2.9 | nM |
Lestaurtinib | TAOK1 | 70.0 | nM |
Lestaurtinib | TAOK2 | 500.0 | nM |
Lestaurtinib | TAOK3 | 86.0 | nM |
Lestaurtinib | TBK1 | 18.0 | nM |
Lestaurtinib | TEC | 1200.0 | nM |
Lestaurtinib | TESK1 | 290.0 | nM |
Lestaurtinib | TGFBR1 | 120.0 | nM |
Lestaurtinib | TGFBR2 | 540.0 | nM |
Lestaurtinib | TIE1 | 680.0 | nM |
Lestaurtinib | TIE2 | 630.0 | nM |
Lestaurtinib | TLK1 | 110.0 | nM |
Lestaurtinib | TLK2 | 64.0 | nM |
Lestaurtinib | TNIK | 5.4 | nM |
Lestaurtinib | TNK1 | 9.3 | nM |
Lestaurtinib | TNK2 | 6.6 | nM |
Lestaurtinib | TNNI3K | 2100.0 | nM |
Lestaurtinib | TRKA | 8.3 | nM |
Lestaurtinib | TRKB | 14.0 | nM |
Lestaurtinib | TRKC | 14.0 | nM |
Lestaurtinib | TRPM6 | nM | |
Lestaurtinib | TSSK1 | 98.0 | nM |
Lestaurtinib | TTK | 6.5 | nM |
Lestaurtinib | TXK | 660.0 | nM |
Lestaurtinib | TYK2(JH1domain-catalytic) | 15.0 | nM |