CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | PRKX | 42.0 | nM |
| Lestaurtinib | PRP4 | 550.0 | nM |
| Lestaurtinib | FAK2 | 41.0 | nM |
| Lestaurtinib | SIK3 | 120.0 | nM |
| Lestaurtinib | RAF1 | nM | |
| Lestaurtinib | RET | 20.0 | nM |
| Lestaurtinib | RET(M918T) | 14.0 | nM |
| Lestaurtinib | RET(V804L) | 6.7 | nM |
| Lestaurtinib | RET(V804M) | 4.7 | nM |
| Lestaurtinib | RIOK1 | 9.0 | nM |
| Lestaurtinib | RIOK2 | 6700.0 | nM |
| Lestaurtinib | RIOK3 | 7.7 | nM |
| Lestaurtinib | RIPK1 | nM | |
| Lestaurtinib | RIPK2 | 640.0 | nM |
| Lestaurtinib | RIPK4 | 13.0 | nM |
| Lestaurtinib | RIPK5 | 5.3 | nM |
| Lestaurtinib | ROCK1 | 56.0 | nM |
| Lestaurtinib | ROCK2 | 71.0 | nM |
| Lestaurtinib | ROS1 | 26.0 | nM |
| Lestaurtinib | RPS6KA4(Kin.Dom.1-N-terminal) | 62.0 | nM |
| Lestaurtinib | RPS6KA4(Kin.Dom.2-C-terminal) | 1300.0 | nM |
| Lestaurtinib | RPS6KA5(Kin.Dom.1-N-terminal) | 42.0 | nM |
| Lestaurtinib | RPS6KA5(Kin.Dom.2-C-terminal) | 960.0 | nM |
| Lestaurtinib | RSK1(Kin.Dom.1-N-terminal) | 28.0 | nM |
| Lestaurtinib | RSK1(Kin.Dom.2-C-terminal) | 2400.0 | nM |