CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | PFCDPK1(P.falciparum) | 5.6 | nM |
| Lestaurtinib | PFPK5(P.falciparum) | 5600.0 | nM |
| Lestaurtinib | CDK15 | 1300.0 | nM |
| Lestaurtinib | CDK14 | 720.0 | nM |
| Lestaurtinib | PHKG1 | 0.4 | nM |
| Lestaurtinib | PHKG2 | 1.7 | nM |
| Lestaurtinib | PIK3C2B | 5200.0 | nM |
| Lestaurtinib | PIK3C2G | 230.0 | nM |
| Lestaurtinib | PIK3CA | 4900.0 | nM |
| Lestaurtinib | PIK3CA(C420R) | 4900.0 | nM |
| Lestaurtinib | PIK3CA(E542K) | 5900.0 | nM |
| Lestaurtinib | PIK3CA(E545A) | 5600.0 | nM |
| Lestaurtinib | PIK3CA(E545K) | 7400.0 | nM |
| Lestaurtinib | PIK3CA(H1047L) | 49.0 | nM |
| Lestaurtinib | PIK3CA(H1047Y) | 650.0 | nM |
| Lestaurtinib | PIK3CA(I800L) | nM | |
| Lestaurtinib | PIK3CA(M1043I) | 1100.0 | nM |
| Lestaurtinib | PIK3CA(Q546K) | 5400.0 | nM |
| Lestaurtinib | PIK3CB | 6700.0 | nM |
| Lestaurtinib | PIK3CD | 4000.0 | nM |
| Lestaurtinib | PIK3CG | 350.0 | nM |
| Lestaurtinib | PIK4CB | 290.0 | nM |
| Lestaurtinib | PIM1 | 200.0 | nM |
| Lestaurtinib | PIM2 | 250.0 | nM |
| Lestaurtinib | PIM3 | 18.0 | nM |