CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | IKKB | 12.0 | nM |
Lestaurtinib | IKKE | 11.0 | nM |
Lestaurtinib | INSR | 1100.0 | nM |
Lestaurtinib | INSRR | 1800.0 | nM |
Lestaurtinib | IRAK1 | 6.1 | nM |
Lestaurtinib | IRAK3 | 16.0 | nM |
Lestaurtinib | IRAK4 | 1.7 | nM |
Lestaurtinib | ITK | 290.0 | nM |
Lestaurtinib | JAK1(JH1domain-catalytic) | 8.8 | nM |
Lestaurtinib | JAK1(JH2domain-pseudokinase) | nM | |
Lestaurtinib | JAK2(JH1domain-catalytic) | 3.7 | nM |
Lestaurtinib | JAK3(JH1domain-catalytic) | 2.3 | nM |
Lestaurtinib | JNK1 | 11.0 | nM |
Lestaurtinib | JNK3 | 12.0 | nM |
Lestaurtinib | KC1G1 | nM | |
Lestaurtinib | KC1G2 | nM | |
Lestaurtinib | KCC2D | 8.8 | nM |
Lestaurtinib | KCC4 | 3000.0 | nM |
Lestaurtinib | KGP1 | 370.0 | nM |
Lestaurtinib | KGP2 | 25.0 | nM |
Lestaurtinib | KIT | 150.0 | nM |
Lestaurtinib | KIT(A829P) | 35.0 | nM |
Lestaurtinib | KIT(D816H) | 11.0 | nM |
Lestaurtinib | KIT(D816V) | 7.1 | nM |
Lestaurtinib | KIT(L576P) | 40.0 | nM |