CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib CAMK2B 59.0
nM
Lestaurtinib CAMK2G 26.0
nM
Lestaurtinib CAMKK2 15.0
nM
Lestaurtinib CASK 330.0
nM
Lestaurtinib CDC2L1
nM
Lestaurtinib CDC2L2
nM
Lestaurtinib CDC2L5 1000.0
nM
Lestaurtinib CDK11
nM
Lestaurtinib CDK14 720.0
nM
Lestaurtinib CDK15 1300.0
nM
Lestaurtinib CDK16 27.0
nM
Lestaurtinib CDK2 20.0
nM
Lestaurtinib CDK3 420.0
nM
Lestaurtinib CDK4-cyclinD1 30.0
nM
Lestaurtinib CDK4-cyclinD3 35.0
nM
Lestaurtinib CDK5 410.0
nM
Lestaurtinib CDK7 87.0
nM
Lestaurtinib CDK8 8000.0
nM
Lestaurtinib CDK9 530.0
nM
Lestaurtinib CDKL1 490.0
nM
Lestaurtinib CDKL2 43.0
nM
Lestaurtinib CDKL3 430.0
nM
Lestaurtinib CDKL5 10.0
nM
Lestaurtinib CHEK1 2.8
nM
Lestaurtinib CHK2 210.0
nM