CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | M3K5 | 70.0 | nM |
Lestaurtinib | ALK | 71.0 | nM |
Lestaurtinib | ROCK2 | 71.0 | nM |
Lestaurtinib | ACVR1 | 75.0 | nM |
Lestaurtinib | KIT(V559D) | 76.0 | nM |
Lestaurtinib | DAPK1 | 80.0 | nM |
Lestaurtinib | MP2K7 | 80.0 | nM |
Lestaurtinib | DAPK3 | 82.0 | nM |
Lestaurtinib | SIK1 | 82.0 | nM |
Lestaurtinib | MARK1 | 83.0 | nM |
Lestaurtinib | FYN | 84.0 | nM |
Lestaurtinib | CIT | 85.0 | nM |
Lestaurtinib | TAOK3 | 86.0 | nM |
Lestaurtinib | ACVR1B | 86.0 | nM |
Lestaurtinib | CDK7 | 87.0 | nM |
Lestaurtinib | RSK3(Kin.Dom.1-N-terminal) | 88.0 | nM |
Lestaurtinib | YSK1 | 97.0 | nM |
Lestaurtinib | TSSK1 | 98.0 | nM |
Lestaurtinib | EPHB6 | 98.0 | nM |
Lestaurtinib | KPCT | 100.0 | nM |
Lestaurtinib | TLK1 | 110.0 | nM |
Lestaurtinib | CSF1R | 110.0 | nM |
Lestaurtinib | RSK4(Kin.Dom.1-N-terminal) | 110.0 | nM |
Lestaurtinib | M4K3 | 110.0 | nM |
Lestaurtinib | PRKR | 120.0 | nM |