CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib M3K5 70.0
nM
Lestaurtinib ALK 71.0
nM
Lestaurtinib ROCK2 71.0
nM
Lestaurtinib ACVR1 75.0
nM
Lestaurtinib KIT(V559D) 76.0
nM
Lestaurtinib DAPK1 80.0
nM
Lestaurtinib MP2K7 80.0
nM
Lestaurtinib DAPK3 82.0
nM
Lestaurtinib SIK1 82.0
nM
Lestaurtinib MARK1 83.0
nM
Lestaurtinib FYN 84.0
nM
Lestaurtinib CIT 85.0
nM
Lestaurtinib TAOK3 86.0
nM
Lestaurtinib ACVR1B 86.0
nM
Lestaurtinib CDK7 87.0
nM
Lestaurtinib RSK3(Kin.Dom.1-N-terminal) 88.0
nM
Lestaurtinib YSK1 97.0
nM
Lestaurtinib TSSK1 98.0
nM
Lestaurtinib EPHB6 98.0
nM
Lestaurtinib KPCT 100.0
nM
Lestaurtinib TLK1 110.0
nM
Lestaurtinib CSF1R 110.0
nM
Lestaurtinib RSK4(Kin.Dom.1-N-terminal) 110.0
nM
Lestaurtinib M4K3 110.0
nM
Lestaurtinib PRKR 120.0
nM