CEP-701 KINOMEscan - Dataset (ID:20189)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | CDKL5 | 10.0 | nM |
Lestaurtinib | JNK1 | 11.0 | nM |
Lestaurtinib | KIT(D816H) | 11.0 | nM |
Lestaurtinib | IKKE | 11.0 | nM |
Lestaurtinib | JNK3 | 12.0 | nM |
Lestaurtinib | MLCK | 12.0 | nM |
Lestaurtinib | GRK4 | 12.0 | nM |
Lestaurtinib | IKKB | 12.0 | nM |
Lestaurtinib | SRPK3 | 13.0 | nM |
Lestaurtinib | MYLK | 13.0 | nM |
Lestaurtinib | RIPK4 | 13.0 | nM |
Lestaurtinib | RET(M918T) | 14.0 | nM |
Lestaurtinib | MARK2 | 14.0 | nM |
Lestaurtinib | TRKB | 14.0 | nM |
Lestaurtinib | KPCD1 | 14.0 | nM |
Lestaurtinib | TRKC | 14.0 | nM |
Lestaurtinib | MLK2 | 15.0 | nM |
Lestaurtinib | CAMKK2 | 15.0 | nM |
Lestaurtinib | TYK2(JH1domain-catalytic) | 15.0 | nM |
Lestaurtinib | SIK2 | 15.0 | nM |
Lestaurtinib | BRSK2 | 16.0 | nM |
Lestaurtinib | EGFR(T790M) | 16.0 | nM |
Lestaurtinib | BIKE | 16.0 | nM |
Lestaurtinib | AURKB | 16.0 | nM |
Lestaurtinib | AURKA | 16.0 | nM |