CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | IRAK1 | 6.1 | nM |
Lestaurtinib | TTK | 6.5 | nM |
Lestaurtinib | TNK2 | 6.6 | nM |
Lestaurtinib | RET(V804L) | 6.7 | nM |
Lestaurtinib | MP2K5 | 7.0 | nM |
Lestaurtinib | FLT3(R834Q) | 7.0 | nM |
Lestaurtinib | KIT(D816V) | 7.1 | nM |
Lestaurtinib | GRK7 | 7.2 | nM |
Lestaurtinib | GAK | 7.3 | nM |
Lestaurtinib | RIOK3 | 7.7 | nM |
Lestaurtinib | EGFR(L858R,T790M) | 7.8 | nM |
Lestaurtinib | KPCD2 | 8.1 | nM |
Lestaurtinib | TRKA | 8.3 | nM |
Lestaurtinib | FLT3 | 8.5 | nM |
Lestaurtinib | KCC2D | 8.8 | nM |
Lestaurtinib | JAK1(JH1domain-catalytic) | 8.8 | nM |
Lestaurtinib | KPCD3 | 8.9 | nM |
Lestaurtinib | RIOK1 | 9.0 | nM |
Lestaurtinib | IKKA | 9.0 | nM |
Lestaurtinib | TNK1 | 9.3 | nM |
Lestaurtinib | SYK | 9.5 | nM |
Lestaurtinib | CLK1 | 9.6 | nM |
Lestaurtinib | PAK6 | 9.9 | nM |
Lestaurtinib | CAMK2A | 10.0 | nM |
Lestaurtinib | CDKL5 | 10.0 | nM |