CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | MLK1 | 3.5 | nM |
Lestaurtinib | MINK | 3.6 | nM |
Lestaurtinib | LRRK2 | 3.6 | nM |
Lestaurtinib | JAK2(JH1domain-catalytic) | 3.7 | nM |
Lestaurtinib | NUAK1 | 3.7 | nM |
Lestaurtinib | MP2K4 | 3.8 | nM |
Lestaurtinib | MP2K2 | 3.9 | nM |
Lestaurtinib | GCN2(Kin.Dom.2,S808G) | 4.1 | nM |
Lestaurtinib | AURKC | 4.1 | nM |
Lestaurtinib | MAP4K2 | 4.7 | nM |
Lestaurtinib | RET(V804M) | 4.7 | nM |
Lestaurtinib | M3K2 | 4.8 | nM |
Lestaurtinib | ERK8 | 4.9 | nM |
Lestaurtinib | ULK3 | 4.9 | nM |
Lestaurtinib | MP2K3 | 5.0 | nM |
Lestaurtinib | DRAK2 | 5.0 | nM |
Lestaurtinib | RIPK5 | 5.3 | nM |
Lestaurtinib | PKN1 | 5.3 | nM |
Lestaurtinib | FLT3(K663Q) | 5.4 | nM |
Lestaurtinib | TNIK | 5.4 | nM |
Lestaurtinib | PFCDPK1(P.falciparum) | 5.6 | nM |
Lestaurtinib | LOK | 5.7 | nM |
Lestaurtinib | ERN1 | 5.7 | nM |
Lestaurtinib | SGK3 | 5.8 | nM |
Lestaurtinib | MAP3K3 | 6.0 | nM |