CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | PIK3CA(Q546K) | 5400.0 | nM |
| Lestaurtinib | ERBB3 | 5500.0 | nM |
| Lestaurtinib | PIK3CA(E545A) | 5600.0 | nM |
| Lestaurtinib | PFPK5(P.falciparum) | 5600.0 | nM |
| Lestaurtinib | NEK5 | 5600.0 | nM |
| Lestaurtinib | YANK2 | 5900.0 | nM |
| Lestaurtinib | PIK3CA(E542K) | 5900.0 | nM |
| Lestaurtinib | EPHA5 | 5900.0 | nM |
| Lestaurtinib | AKT3 | 6200.0 | nM |
| Lestaurtinib | ABL2 | 6500.0 | nM |
| Lestaurtinib | RIOK2 | 6700.0 | nM |
| Lestaurtinib | PIK3CB | 6700.0 | nM |
| Lestaurtinib | MLTK | 6700.0 | nM |
| Lestaurtinib | EPHB2 | 6900.0 | nM |
| Lestaurtinib | EPHB4 | 6900.0 | nM |
| Lestaurtinib | CSNK1A1L | 7100.0 | nM |
| Lestaurtinib | PIK3CA(E545K) | 7400.0 | nM |
| Lestaurtinib | ABL1(F317L)-nonphosphorylated | 7600.0 | nM |
| Lestaurtinib | WEE2 | 7900.0 | nM |
| Lestaurtinib | CDK8 | 8000.0 | nM |
| Lestaurtinib | OSR1 | 8000.0 | nM |
| Lestaurtinib | YANK3 | 8000.0 | nM |
| Lestaurtinib | MST1R | 8200.0 | nM |
| Lestaurtinib | RSK4(Kin.Dom.2-C-terminal) | 9100.0 | nM |
| Lestaurtinib | MRCKA | 9200.0 | nM |