CEP-701 KINOMEscan - Dataset (ID:20189)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | TYK2(JH2domain-pseudokinase) | 910.0 | nM |
Lestaurtinib | ABL1(Y253F)-phosphorylated | 910.0 | nM |
Lestaurtinib | MAPKAPK5 | 930.0 | nM |
Lestaurtinib | ABL1(T315I)-nonphosphorylated | 950.0 | nM |
Lestaurtinib | BMPR1A | 950.0 | nM |
Lestaurtinib | RPS6KA5(Kin.Dom.2-C-terminal) | 960.0 | nM |
Lestaurtinib | CSNK2A2 | 970.0 | nM |
Lestaurtinib | CTK | 970.0 | nM |
Lestaurtinib | CDC2L5 | 1000.0 | nM |
Lestaurtinib | MRCKB | 1000.0 | nM |
Lestaurtinib | ULK1 | 1000.0 | nM |
Lestaurtinib | ABL1(H396P)-nonphosphorylated | 1000.0 | nM |
Lestaurtinib | ABL1-phosphorylated | 1000.0 | nM |
Lestaurtinib | EGFR(G719S) | 1100.0 | nM |
Lestaurtinib | EGFR | 1100.0 | nM |
Lestaurtinib | STK39 | 1100.0 | nM |
Lestaurtinib | ERK5 | 1100.0 | nM |
Lestaurtinib | FAK1 | 1100.0 | nM |
Lestaurtinib | PIK3CA(M1043I) | 1100.0 | nM |
Lestaurtinib | INSR | 1100.0 | nM |
Lestaurtinib | DCAMKL3 | 1100.0 | nM |
Lestaurtinib | RSK3(Kin.Dom.2-C-terminal) | 1200.0 | nM |
Lestaurtinib | EPHA6 | 1200.0 | nM |
Lestaurtinib | TEC | 1200.0 | nM |
Lestaurtinib | EGFR(G719C) | 1200.0 | nM |