CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib KGP1 370.0
nM
Lestaurtinib FES 370.0
nM
Lestaurtinib HIPK2 370.0
nM
Lestaurtinib NDR2 370.0
nM
Lestaurtinib EPHA1 380.0
nM
Lestaurtinib KIT(V559D,V654A) 380.0
nM
Lestaurtinib EGFR(E746-A750del) 400.0
nM
Lestaurtinib DDR2 400.0
nM
Lestaurtinib CDK5 410.0
nM
Lestaurtinib CDK3 420.0
nM
Lestaurtinib CDKL3 430.0
nM
Lestaurtinib LCK 430.0
nM
Lestaurtinib CAMK1G 470.0
nM
Lestaurtinib MET(M1250T) 480.0
nM
Lestaurtinib LTK 490.0
nM
Lestaurtinib CDKL1 490.0
nM
Lestaurtinib TAOK2 500.0
nM
Lestaurtinib DDR1 510.0
nM
Lestaurtinib CDK9 530.0
nM
Lestaurtinib TGFBR2 540.0
nM
Lestaurtinib PRP4 550.0
nM
Lestaurtinib EGFR(L747-T751del,Sins) 560.0
nM
Lestaurtinib HUNK 570.0
nM
Lestaurtinib FGFR3 580.0
nM
Lestaurtinib HIPK1 590.0
nM