CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | KGP1 | 370.0 | nM |
Lestaurtinib | FES | 370.0 | nM |
Lestaurtinib | HIPK2 | 370.0 | nM |
Lestaurtinib | NDR2 | 370.0 | nM |
Lestaurtinib | EPHA1 | 380.0 | nM |
Lestaurtinib | KIT(V559D,V654A) | 380.0 | nM |
Lestaurtinib | EGFR(E746-A750del) | 400.0 | nM |
Lestaurtinib | DDR2 | 400.0 | nM |
Lestaurtinib | CDK5 | 410.0 | nM |
Lestaurtinib | CDK3 | 420.0 | nM |
Lestaurtinib | CDKL3 | 430.0 | nM |
Lestaurtinib | LCK | 430.0 | nM |
Lestaurtinib | CAMK1G | 470.0 | nM |
Lestaurtinib | MET(M1250T) | 480.0 | nM |
Lestaurtinib | LTK | 490.0 | nM |
Lestaurtinib | CDKL1 | 490.0 | nM |
Lestaurtinib | TAOK2 | 500.0 | nM |
Lestaurtinib | DDR1 | 510.0 | nM |
Lestaurtinib | CDK9 | 530.0 | nM |
Lestaurtinib | TGFBR2 | 540.0 | nM |
Lestaurtinib | PRP4 | 550.0 | nM |
Lestaurtinib | EGFR(L747-T751del,Sins) | 560.0 | nM |
Lestaurtinib | HUNK | 570.0 | nM |
Lestaurtinib | FGFR3 | 580.0 | nM |
Lestaurtinib | HIPK1 | 590.0 | nM |