CEP-701 KINOMEscan - Dataset (ID:20189)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | ABL2 | 6500.0 | nM |
Lestaurtinib | ABL1(Y253F)-phosphorylated | 910.0 | nM |
Lestaurtinib | ABL1(T315I)-phosphorylated | 160.0 | nM |
Lestaurtinib | ABL1(T315I)-nonphosphorylated | 950.0 | nM |
Lestaurtinib | ABL1(Q252H)-phosphorylated | 830.0 | nM |
Lestaurtinib | ABL1(Q252H)-nonphosphorylated | 2500.0 | nM |
Lestaurtinib | ABL1-phosphorylated | 1000.0 | nM |
Lestaurtinib | ABL1-nonphosphorylated | 3200.0 | nM |
Lestaurtinib | ABL1(M351T)-phosphorylated | 780.0 | nM |
Lestaurtinib | ABL1(H396P)-phosphorylated | 870.0 | nM |
Lestaurtinib | ABL1(H396P)-nonphosphorylated | 1000.0 | nM |
Lestaurtinib | ABL1(F317L)-phosphorylated | 2200.0 | nM |
Lestaurtinib | ABL1(F317L)-nonphosphorylated | 7600.0 | nM |
Lestaurtinib | ABL1(F317I)-phosphorylated | 4900.0 | nM |
Lestaurtinib | ABL1(F317I)-nonphosphorylated | nM | |
Lestaurtinib | ABL1(E255K)-phosphorylated | 840.0 | nM |
Lestaurtinib | AAK1 | 3.1 | nM |