CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | ABL1(Q252H)-nonphosphorylated | 2500.0 | nM |
| Lestaurtinib | ACVR2A | 2500.0 | nM |
| Lestaurtinib | RSK1(Kin.Dom.2-C-terminal) | 2400.0 | nM |
| Lestaurtinib | PLK3 | 2300.0 | nM |
| Lestaurtinib | GSK3A | 2300.0 | nM |
| Lestaurtinib | ABL1(F317L)-phosphorylated | 2200.0 | nM |
| Lestaurtinib | ACVRL1 | 2200.0 | nM |
| Lestaurtinib | AKT2 | 2100.0 | nM |
| Lestaurtinib | TNNI3K | 2100.0 | nM |
| Lestaurtinib | YANK1 | 2100.0 | nM |
| Lestaurtinib | NIM1 | 1800.0 | nM |
| Lestaurtinib | INSRR | 1800.0 | nM |
| Lestaurtinib | KPCI | 1800.0 | nM |
| Lestaurtinib | FGFR4 | 1800.0 | nM |
| Lestaurtinib | EPHA4 | 1700.0 | nM |
| Lestaurtinib | PTK6 | 1700.0 | nM |
| Lestaurtinib | MAK | 1700.0 | nM |
| Lestaurtinib | LIMK1 | 1600.0 | nM |
| Lestaurtinib | BMPR2 | 1500.0 | nM |
| Lestaurtinib | ERBB4 | 1400.0 | nM |
| Lestaurtinib | EGFR(S752-I759del) | 1400.0 | nM |
| Lestaurtinib | EGFR(L747-S752del, P753S) | 1400.0 | nM |
| Lestaurtinib | RPS6KA4(Kin.Dom.2-C-terminal) | 1300.0 | nM |
| Lestaurtinib | CDK15 | 1300.0 | nM |
| Lestaurtinib | GSK3B | 1300.0 | nM |