CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | NEK9 | 5400.0 | nM |
Lestaurtinib | PIK3CA(Q546K) | 5400.0 | nM |
Lestaurtinib | PIK3C2B | 5200.0 | nM |
Lestaurtinib | EPHB1 | 5200.0 | nM |
Lestaurtinib | NEK2 | 4900.0 | nM |
Lestaurtinib | PIK3CA(C420R) | 4900.0 | nM |
Lestaurtinib | PIK3CA | 4900.0 | nM |
Lestaurtinib | ABL1(F317I)-phosphorylated | 4900.0 | nM |
Lestaurtinib | DCAMKL2 | 4500.0 | nM |
Lestaurtinib | NEK6 | 4400.0 | nM |
Lestaurtinib | AKT1 | 4400.0 | nM |
Lestaurtinib | MAP3K1 | 4400.0 | nM |
Lestaurtinib | IGF1R | 4200.0 | nM |
Lestaurtinib | MUSK | 4100.0 | nM |
Lestaurtinib | PIK3CD | 4000.0 | nM |
Lestaurtinib | NEK7 | 4000.0 | nM |
Lestaurtinib | STK36 | 3800.0 | nM |
Lestaurtinib | ACVR2B | 3800.0 | nM |
Lestaurtinib | MK13 | 3500.0 | nM |
Lestaurtinib | ABL1-nonphosphorylated | 3200.0 | nM |
Lestaurtinib | KCC4 | 3000.0 | nM |
Lestaurtinib | MAP3K4 | 2600.0 | nM |
Lestaurtinib | CSNK2A1 | 2600.0 | nM |
Lestaurtinib | DMPK2 | 2500.0 | nM |
Lestaurtinib | ABL1(Q252H)-nonphosphorylated | 2500.0 | nM |