CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | PAK2 | 43.0 | nM |
Lestaurtinib | CDKL2 | 43.0 | nM |
Lestaurtinib | PRKX | 42.0 | nM |
Lestaurtinib | RPS6KA5(Kin.Dom.1-N-terminal) | 42.0 | nM |
Lestaurtinib | FAK2 | 41.0 | nM |
Lestaurtinib | MET(Y1235D) | 41.0 | nM |
Lestaurtinib | KIT(L576P) | 40.0 | nM |
Lestaurtinib | ICK | 39.0 | nM |
Lestaurtinib | M4K1 | 38.0 | nM |
Lestaurtinib | PIP5K1A | 36.0 | nM |
Lestaurtinib | CDK4-cyclinD3 | 35.0 | nM |
Lestaurtinib | AXL | 35.0 | nM |
Lestaurtinib | KIT(A829P) | 35.0 | nM |
Lestaurtinib | PAK3 | 35.0 | nM |
Lestaurtinib | SLK | 35.0 | nM |
Lestaurtinib | ANKK1 | 32.0 | nM |
Lestaurtinib | MERTK | 32.0 | nM |
Lestaurtinib | PAK1 | 30.0 | nM |
Lestaurtinib | LATS1 | 30.0 | nM |
Lestaurtinib | CDK4-cyclinD1 | 30.0 | nM |
Lestaurtinib | PGFRB | 29.0 | nM |
Lestaurtinib | DYRK1B | 29.0 | nM |
Lestaurtinib | MYLK4 | 29.0 | nM |
Lestaurtinib | FER | 28.0 | nM |
Lestaurtinib | RSK1(Kin.Dom.1-N-terminal) | 28.0 | nM |