CEP-701 KINOMEscan - Dataset (ID:20189)

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Small Molecule Protein Kd Conc unit
Lestaurtinib PAK2 43.0
nM
Lestaurtinib CDKL2 43.0
nM
Lestaurtinib PRKX 42.0
nM
Lestaurtinib RPS6KA5(Kin.Dom.1-N-terminal) 42.0
nM
Lestaurtinib FAK2 41.0
nM
Lestaurtinib MET(Y1235D) 41.0
nM
Lestaurtinib KIT(L576P) 40.0
nM
Lestaurtinib ICK 39.0
nM
Lestaurtinib M4K1 38.0
nM
Lestaurtinib PIP5K1A 36.0
nM
Lestaurtinib CDK4-cyclinD3 35.0
nM
Lestaurtinib AXL 35.0
nM
Lestaurtinib KIT(A829P) 35.0
nM
Lestaurtinib PAK3 35.0
nM
Lestaurtinib SLK 35.0
nM
Lestaurtinib ANKK1 32.0
nM
Lestaurtinib MERTK 32.0
nM
Lestaurtinib PAK1 30.0
nM
Lestaurtinib LATS1 30.0
nM
Lestaurtinib CDK4-cyclinD1 30.0
nM
Lestaurtinib PGFRB 29.0
nM
Lestaurtinib DYRK1B 29.0
nM
Lestaurtinib MYLK4 29.0
nM
Lestaurtinib FER 28.0
nM
Lestaurtinib RSK1(Kin.Dom.1-N-terminal) 28.0
nM