CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | FES | 370.0 | nM |
| Lestaurtinib | FGFR1 | 310.0 | nM |
| Lestaurtinib | FGFR2 | 660.0 | nM |
| Lestaurtinib | FGFR3 | 580.0 | nM |
| Lestaurtinib | FGFR3(G697C) | 730.0 | nM |
| Lestaurtinib | FGFR4 | 1800.0 | nM |
| Lestaurtinib | FGR | 52.0 | nM |
| Lestaurtinib | VGFR1 | 120.0 | nM |
| Lestaurtinib | FLT3 | 8.5 | nM |
| Lestaurtinib | FLT3(D835H) | 0.7 | nM |
| Lestaurtinib | FLT3(D835Y) | 0.6 | nM |
| Lestaurtinib | FLT3(ITD) | 1.5 | nM |
| Lestaurtinib | FLT3(K663Q) | 5.4 | nM |
| Lestaurtinib | FLT3(N841I) | 1.4 | nM |
| Lestaurtinib | FLT3(R834Q) | 7.0 | nM |
| Lestaurtinib | FLT4 | 17.0 | nM |
| Lestaurtinib | FRK | 740.0 | nM |
| Lestaurtinib | FYN | 84.0 | nM |
| Lestaurtinib | GAK | 7.3 | nM |
| Lestaurtinib | GCN2(Kin.Dom.2,S808G) | 4.1 | nM |
| Lestaurtinib | GRK1 | 24.0 | nM |
| Lestaurtinib | GRK4 | 12.0 | nM |
| Lestaurtinib | GRK7 | 7.2 | nM |
| Lestaurtinib | GSK3A | 2300.0 | nM |
| Lestaurtinib | GSK3B | 1300.0 | nM |