CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Lestaurtinib | DCAMKL2 | 4500.0 | nM |
| Lestaurtinib | DCAMKL3 | 1100.0 | nM |
| Lestaurtinib | DDR1 | 510.0 | nM |
| Lestaurtinib | DDR2 | 400.0 | nM |
| Lestaurtinib | M3K12 | 840.0 | nM |
| Lestaurtinib | DMPK | 240.0 | nM |
| Lestaurtinib | DMPK2 | 2500.0 | nM |
| Lestaurtinib | DRAK1 | 3.4 | nM |
| Lestaurtinib | DRAK2 | 5.0 | nM |
| Lestaurtinib | DYRK1A | 20.0 | nM |
| Lestaurtinib | DYRK1B | 29.0 | nM |
| Lestaurtinib | DYRK2 | 22.0 | nM |
| Lestaurtinib | EGFR | 1100.0 | nM |
| Lestaurtinib | EGFR(E746-A750del) | 400.0 | nM |
| Lestaurtinib | EGFR(G719C) | 1200.0 | nM |
| Lestaurtinib | EGFR(G719S) | 1100.0 | nM |
| Lestaurtinib | EGFR(L747-E749del, A750P) | 320.0 | nM |
| Lestaurtinib | EGFR(L747-S752del, P753S) | 1400.0 | nM |
| Lestaurtinib | EGFR(L747-T751del,Sins) | 560.0 | nM |
| Lestaurtinib | EGFR(L858R) | 860.0 | nM |
| Lestaurtinib | EGFR(L858R,T790M) | 7.8 | nM |
| Lestaurtinib | EGFR(L861Q) | 800.0 | nM |
| Lestaurtinib | EGFR(S752-I759del) | 1400.0 | nM |
| Lestaurtinib | EGFR(T790M) | 16.0 | nM |
| Lestaurtinib | EIF2AK1 | nM |