CEP-701 KINOMEscan - Dataset (ID:20189)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Lestaurtinib | RSK2(Kin.Dom.1-N-terminal) | 290.0 | nM |
Lestaurtinib | RSK3(Kin.Dom.1-N-terminal) | 88.0 | nM |
Lestaurtinib | RSK3(Kin.Dom.2-C-terminal) | 1200.0 | nM |
Lestaurtinib | RSK4(Kin.Dom.1-N-terminal) | 110.0 | nM |
Lestaurtinib | RSK4(Kin.Dom.2-C-terminal) | 9100.0 | nM |
Lestaurtinib | S6K1 | 69.0 | nM |
Lestaurtinib | SBK1 | 200.0 | nM |
Lestaurtinib | SgK110 | 120.0 | nM |
Lestaurtinib | SGK3 | 5.8 | nM |
Lestaurtinib | SIK1 | 82.0 | nM |
Lestaurtinib | SIK2 | 15.0 | nM |
Lestaurtinib | SLK | 35.0 | nM |
Lestaurtinib | SNARK | 1.0 | nM |
Lestaurtinib | SNRK | nM | |
Lestaurtinib | SRC | 640.0 | nM |
Lestaurtinib | SRMS | 820.0 | nM |
Lestaurtinib | SRPK1 | 10.0 | nM |
Lestaurtinib | SRPK2 | 51.0 | nM |
Lestaurtinib | SRPK3 | 13.0 | nM |
Lestaurtinib | STK16 | 19.0 | nM |
Lestaurtinib | STK33 | 26.0 | nM |
Lestaurtinib | STK35 | 810.0 | nM |
Lestaurtinib | STK36 | 3800.0 | nM |
Lestaurtinib | STK39 | 1100.0 | nM |
Lestaurtinib | SYK | 9.5 | nM |