CP-690550 KINOMEscan - Dataset (ID:20188)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tofacitinib | PRKX | nM | |
| Tofacitinib | PRP4 | nM | |
| Tofacitinib | FAK2 | nM | |
| Tofacitinib | SIK3 | nM | |
| Tofacitinib | RAF1 | nM | |
| Tofacitinib | RET | nM | |
| Tofacitinib | RET(M918T) | 3300.0 | nM |
| Tofacitinib | RET(V804L) | nM | |
| Tofacitinib | RET(V804M) | nM | |
| Tofacitinib | RIOK1 | nM | |
| Tofacitinib | RIOK2 | nM | |
| Tofacitinib | RIOK3 | nM | |
| Tofacitinib | RIPK1 | nM | |
| Tofacitinib | RIPK2 | nM | |
| Tofacitinib | RIPK4 | nM | |
| Tofacitinib | RIPK5 | nM | |
| Tofacitinib | ROCK1 | 470.0 | nM |
| Tofacitinib | ROCK2 | 420.0 | nM |
| Tofacitinib | ROS1 | nM | |
| Tofacitinib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
| Tofacitinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
| Tofacitinib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
| Tofacitinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
| Tofacitinib | RSK1(Kin.Dom.1-N-terminal) | nM | |
| Tofacitinib | RSK1(Kin.Dom.2-C-terminal) | 1400.0 | nM |