CP-690550 KINOMEscan - Dataset (ID:20188)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tofacitinib | IKKB | nM | |
Tofacitinib | IKKE | nM | |
Tofacitinib | INSR | nM | |
Tofacitinib | INSRR | nM | |
Tofacitinib | IRAK1 | nM | |
Tofacitinib | IRAK3 | nM | |
Tofacitinib | IRAK4 | nM | |
Tofacitinib | ITK | nM | |
Tofacitinib | JAK1(JH1domain-catalytic) | 1.6 | nM |
Tofacitinib | JAK1(JH2domain-pseudokinase) | nM | |
Tofacitinib | JAK2(JH1domain-catalytic) | 0.6 | nM |
Tofacitinib | JAK3(JH1domain-catalytic) | 0.2 | nM |
Tofacitinib | JNK1 | nM | |
Tofacitinib | JNK3 | nM | |
Tofacitinib | KC1G1 | nM | |
Tofacitinib | KC1G2 | nM | |
Tofacitinib | KCC2D | 2700.0 | nM |
Tofacitinib | KCC4 | nM | |
Tofacitinib | KGP1 | nM | |
Tofacitinib | KGP2 | nM | |
Tofacitinib | KIT | nM | |
Tofacitinib | KIT(A829P) | nM | |
Tofacitinib | KIT(D816H) | nM | |
Tofacitinib | KIT(D816V) | nM | |
Tofacitinib | KIT(L576P) | nM |