CP-690550 KINOMEscan - Dataset (ID:20188)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tofacitinib | KCC2D | 2700.0 | nM |
Tofacitinib | RET(M918T) | 3300.0 | nM |
Tofacitinib | CAMK2A | 3500.0 | nM |
Tofacitinib | GRK7 | 4300.0 | nM |
Tofacitinib | ABL1(H396P)-nonphosphorylated | 4500.0 | nM |
Tofacitinib | MAP4K2 | 4800.0 | nM |
Tofacitinib | ULK3 | 6400.0 | nM |
Tofacitinib | DCLK1 | 6700.0 | nM |
Tofacitinib | ABL1(H396P)-phosphorylated | 6700.0 | nM |
Tofacitinib | BIKE | 7100.0 | nM |
Tofacitinib | ANKK1 | nM | |
Tofacitinib | AMPK-alpha2 | nM | |
Tofacitinib | ABL1-nonphosphorylated | nM | |
Tofacitinib | AMPK-alpha1 | nM | |
Tofacitinib | ALK | nM | |
Tofacitinib | ABL1(Y253F)-phosphorylated | nM | |
Tofacitinib | AKT3 | nM | |
Tofacitinib | AKT2 | nM | |
Tofacitinib | AKT1 | nM | |
Tofacitinib | BRSK2 | nM | |
Tofacitinib | BRSK1 | nM | |
Tofacitinib | ADCK4 | nM | |
Tofacitinib | ABL1(T315I)-nonphosphorylated | nM | |
Tofacitinib | ABL1(F317L)-phosphorylated | nM | |
Tofacitinib | ABL1(F317I)-nonphosphorylated | nM |