CP-690550 KINOMEscan - Dataset (ID:20188)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tofacitinib | LCK | 460.0 | nM |
Tofacitinib | ROCK2 | 420.0 | nM |
Tofacitinib | SNARK | 240.0 | nM |
Tofacitinib | PKN1 | 170.0 | nM |
Tofacitinib | TNK1 | 120.0 | nM |
Tofacitinib | DCAMKL3 | 12.0 | nM |
Tofacitinib | TYK2(JH1domain-catalytic) | 4.8 | nM |
Tofacitinib | JAK1(JH1domain-catalytic) | 1.6 | nM |
Tofacitinib | JAK2(JH1domain-catalytic) | 0.6 | nM |
Tofacitinib | JAK3(JH1domain-catalytic) | 0.2 | nM |
Tofacitinib | ANKK1 | nM | |
Tofacitinib | AMPK-alpha2 | nM | |
Tofacitinib | ABL1-nonphosphorylated | nM | |
Tofacitinib | AMPK-alpha1 | nM | |
Tofacitinib | ALK | nM | |
Tofacitinib | ABL1(Y253F)-phosphorylated | nM | |
Tofacitinib | AKT3 | nM | |
Tofacitinib | AKT2 | nM | |
Tofacitinib | AKT1 | nM | |
Tofacitinib | BRSK2 | nM | |
Tofacitinib | BRSK1 | nM | |
Tofacitinib | ADCK4 | nM | |
Tofacitinib | ABL1(T315I)-nonphosphorylated | nM | |
Tofacitinib | ABL1(F317L)-phosphorylated | nM | |
Tofacitinib | ABL1(F317I)-nonphosphorylated | nM |