PKC-412 KINOMEscan - Dataset (ID:20187)

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Small Molecule Protein Kd Conc unit
PKC412 KIT 220.0
nM
PKC412 KIT(A829P) 43.0
nM
PKC412 KIT(D816H) 16.0
nM
PKC412 KIT(D816V) 7.7
nM
PKC412 KIT(L576P) 41.0
nM
PKC412 KIT(V559D) 200.0
nM
PKC412 KIT(V559D,T670I) 150.0
nM
PKC412 KIT(V559D,V654A) 1600.0
nM
PKC412 LATS1 1100.0
nM
PKC412 LATS2 2200.0
nM
PKC412 LCK 280.0
nM
PKC412 LIMK1
nM
PKC412 LIMK2
nM
PKC412 LKB1 350.0
nM
PKC412 LOK 590.0
nM
PKC412 LRRK2 570.0
nM
PKC412 LRRK2(G2019S) 180.0
nM
PKC412 LTK 3000.0
nM
PKC412 LYN 4200.0
nM
PKC412 M3K13 2800.0
nM
PKC412 MAK
nM
PKC412 MAP3K1
nM
PKC412 MAP3K15
nM
PKC412 M3K2 140.0
nM
PKC412 MAP3K3 210.0
nM