PKC-412 KINOMEscan - Dataset (ID:20187)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PKC412 | KIT | 220.0 | nM |
PKC412 | KIT(A829P) | 43.0 | nM |
PKC412 | KIT(D816H) | 16.0 | nM |
PKC412 | KIT(D816V) | 7.7 | nM |
PKC412 | KIT(L576P) | 41.0 | nM |
PKC412 | KIT(V559D) | 200.0 | nM |
PKC412 | KIT(V559D,T670I) | 150.0 | nM |
PKC412 | KIT(V559D,V654A) | 1600.0 | nM |
PKC412 | LATS1 | 1100.0 | nM |
PKC412 | LATS2 | 2200.0 | nM |
PKC412 | LCK | 280.0 | nM |
PKC412 | LIMK1 | nM | |
PKC412 | LIMK2 | nM | |
PKC412 | LKB1 | 350.0 | nM |
PKC412 | LOK | 590.0 | nM |
PKC412 | LRRK2 | 570.0 | nM |
PKC412 | LRRK2(G2019S) | 180.0 | nM |
PKC412 | LTK | 3000.0 | nM |
PKC412 | LYN | 4200.0 | nM |
PKC412 | M3K13 | 2800.0 | nM |
PKC412 | MAK | nM | |
PKC412 | MAP3K1 | nM | |
PKC412 | MAP3K15 | nM | |
PKC412 | M3K2 | 140.0 | nM |
PKC412 | MAP3K3 | 210.0 | nM |