PKC-412 KINOMEscan - Dataset (ID:20187)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PKC412 | FES | nM | |
PKC412 | FGFR1 | 1600.0 | nM |
PKC412 | FGFR2 | 2400.0 | nM |
PKC412 | FGFR3 | 1700.0 | nM |
PKC412 | FGFR3(G697C) | nM | |
PKC412 | FGFR4 | nM | |
PKC412 | FGR | 730.0 | nM |
PKC412 | VGFR1 | 450.0 | nM |
PKC412 | FLT3 | 11.0 | nM |
PKC412 | FLT3(D835H) | 6.8 | nM |
PKC412 | FLT3(D835Y) | 15.0 | nM |
PKC412 | FLT3(ITD) | 11.0 | nM |
PKC412 | FLT3(K663Q) | 2.0 | nM |
PKC412 | FLT3(N841I) | 6.0 | nM |
PKC412 | FLT3(R834Q) | 12.0 | nM |
PKC412 | FLT4 | 670.0 | nM |
PKC412 | FRK | 2400.0 | nM |
PKC412 | FYN | 2100.0 | nM |
PKC412 | GAK | 380.0 | nM |
PKC412 | GCN2(Kin.Dom.2,S808G) | 39.0 | nM |
PKC412 | GRK1 | 85.0 | nM |
PKC412 | GRK4 | 110.0 | nM |
PKC412 | GRK7 | 48.0 | nM |
PKC412 | GSK3A | 2500.0 | nM |
PKC412 | GSK3B | 1800.0 | nM |