Vandetanib KINOMEscan - Dataset (ID:20186)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Vandetanib | DCAMKL2 | nM | |
Vandetanib | DCAMKL3 | nM | |
Vandetanib | DDR1 | 11.0 | nM |
Vandetanib | DDR2 | 320.0 | nM |
Vandetanib | M3K12 | nM | |
Vandetanib | DMPK | nM | |
Vandetanib | DMPK2 | 2200.0 | nM |
Vandetanib | DRAK1 | nM | |
Vandetanib | DRAK2 | nM | |
Vandetanib | DYRK1A | nM | |
Vandetanib | DYRK1B | nM | |
Vandetanib | DYRK2 | nM | |
Vandetanib | EGFR | 9.5 | nM |
Vandetanib | EGFR(E746-A750del) | 4.8 | nM |
Vandetanib | EGFR(G719C) | 9.6 | nM |
Vandetanib | EGFR(G719S) | 5.9 | nM |
Vandetanib | EGFR(L747-E749del, A750P) | 12.0 | nM |
Vandetanib | EGFR(L747-S752del, P753S) | 7.9 | nM |
Vandetanib | EGFR(L747-T751del,Sins) | 8.9 | nM |
Vandetanib | EGFR(L858R) | 8.7 | nM |
Vandetanib | EGFR(L858R,T790M) | 230.0 | nM |
Vandetanib | EGFR(L861Q) | 11.0 | nM |
Vandetanib | EGFR(S752-I759del) | 12.0 | nM |
Vandetanib | EGFR(T790M) | 100.0 | nM |
Vandetanib | EIF2AK1 | nM |