SKI-606 KINOMEscan - Dataset (ID:20184)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | ABL1(F317L)-phosphorylated | 0.03 | nM |
Bosutinib | ABL1(Y253F)-phosphorylated | 0.04 | nM |
Bosutinib | ABL1(Q252H)-phosphorylated | 0.04 | nM |
Bosutinib | ABL1(M351T)-phosphorylated | 0.04 | nM |
Bosutinib | ABL1(E255K)-phosphorylated | 0.05 | nM |
Bosutinib | ABL1(H396P)-nonphosphorylated | 0.06 | nM |
Bosutinib | ABL1-phosphorylated | 0.06 | nM |
Bosutinib | ABL1(H396P)-phosphorylated | 0.06 | nM |
Bosutinib | ABL1(Q252H)-nonphosphorylated | 0.09 | nM |
Bosutinib | ABL1(F317L)-nonphosphorylated | 0.11 | nM |
Bosutinib | ABL1-nonphosphorylated | 0.12 | nM |
Bosutinib | ABL1(F317I)-phosphorylated | 0.18 | nM |
Bosutinib | MAP4K5 | 0.50 | nM |
Bosutinib | LCK | 0.59 | nM |
Bosutinib | ABL1(F317I)-nonphosphorylated | 0.63 | nM |
Bosutinib | ERBB3 | 0.77 | nM |
Bosutinib | SRC | 1.00 | nM |
Bosutinib | GAK | 1.30 | nM |
Bosutinib | FRK | 1.40 | nM |
Bosutinib | ABL2 | 1.50 | nM |
Bosutinib | STK35 | 2.00 | nM |
Bosutinib | MAP4K2 | 3.10 | nM |
Bosutinib | MINK | 3.20 | nM |
Bosutinib | BLK | 3.30 | nM |
Bosutinib | HCK | 3.40 | nM |