SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | EGFR(G719S) | 26.00 | nM |
Bosutinib | EPHA5 | 27.00 | nM |
Bosutinib | TNK2 | 29.00 | nM |
Bosutinib | EGFR(L747-E749del, A750P) | 29.00 | nM |
Bosutinib | SIK2 | 29.00 | nM |
Bosutinib | EGFR(L747-T751del,Sins) | 30.00 | nM |
Bosutinib | SIK1 | 30.00 | nM |
Bosutinib | M3K2 | 30.00 | nM |
Bosutinib | TNIK | 31.00 | nM |
Bosutinib | CSK | 32.00 | nM |
Bosutinib | EPHB1 | 33.00 | nM |
Bosutinib | EGFR | 35.00 | nM |
Bosutinib | MST4 | 37.00 | nM |
Bosutinib | STK33 | 37.00 | nM |
Bosutinib | EGFR(L747-S752del, P753S) | 38.00 | nM |
Bosutinib | AXL | 52.00 | nM |
Bosutinib | IKKE | 53.00 | nM |
Bosutinib | MAP3K3 | 54.00 | nM |
Bosutinib | TYRO3 | 61.00 | nM |
Bosutinib | SIK3 | 64.00 | nM |
Bosutinib | EGFR(L861Q) | 71.00 | nM |
Bosutinib | TXK | 72.00 | nM |
Bosutinib | KIT(D816V) | 73.00 | nM |
Bosutinib | MLTK | 80.00 | nM |
Bosutinib | DMPK | 91.00 | nM |