SKI-606 KINOMEscan - Dataset (ID:20184)

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Small Molecule Protein Kd Conc unit
Bosutinib EGFR(G719S) 26.00
nM
Bosutinib EPHA5 27.00
nM
Bosutinib TNK2 29.00
nM
Bosutinib EGFR(L747-E749del, A750P) 29.00
nM
Bosutinib SIK2 29.00
nM
Bosutinib EGFR(L747-T751del,Sins) 30.00
nM
Bosutinib SIK1 30.00
nM
Bosutinib M3K2 30.00
nM
Bosutinib TNIK 31.00
nM
Bosutinib CSK 32.00
nM
Bosutinib EPHB1 33.00
nM
Bosutinib EGFR 35.00
nM
Bosutinib MST4 37.00
nM
Bosutinib STK33 37.00
nM
Bosutinib EGFR(L747-S752del, P753S) 38.00
nM
Bosutinib AXL 52.00
nM
Bosutinib IKKE 53.00
nM
Bosutinib MAP3K3 54.00
nM
Bosutinib TYRO3 61.00
nM
Bosutinib SIK3 64.00
nM
Bosutinib EGFR(L861Q) 71.00
nM
Bosutinib TXK 72.00
nM
Bosutinib KIT(D816V) 73.00
nM
Bosutinib MLTK 80.00
nM
Bosutinib DMPK 91.00
nM