SKI-606 KINOMEscan - Dataset (ID:20184)

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Small Molecule Protein Kd Conc unit
Bosutinib ABL1(T315I)-phosphorylated 3.60
nM
Bosutinib YES 4.00
nM
Bosutinib LYN 4.20
nM
Bosutinib SLK 4.70
nM
Bosutinib BTK 4.80
nM
Bosutinib M4K3 5.10
nM
Bosutinib EPHA3 5.80
nM
Bosutinib FGR 6.30
nM
Bosutinib LOK 7.00
nM
Bosutinib MP2K5 8.20
nM
Bosutinib MAP4K4 8.20
nM
Bosutinib EPHB2 8.40
nM
Bosutinib EPHA8 9.00
nM
Bosutinib EPHB4 9.20
nM
Bosutinib MP2K2 9.90
nM
Bosutinib FYN 11.00
nM
Bosutinib M4K1 15.00
nM
Bosutinib YSK4 16.00
nM
Bosutinib EPHA4 18.00
nM
Bosutinib EGFR(E746-A750del) 18.00
nM
Bosutinib EPHA2 18.00
nM
Bosutinib MP2K1 19.00
nM
Bosutinib ABL1(T315I)-nonphosphorylated 21.00
nM
Bosutinib EGFR(L858R) 23.00
nM
Bosutinib ERBB4 26.00
nM