SKI-606 KINOMEscan - Dataset (ID:20184)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Bosutinib | ABL1(T315I)-phosphorylated | 3.60 | nM |
Bosutinib | YES | 4.00 | nM |
Bosutinib | LYN | 4.20 | nM |
Bosutinib | SLK | 4.70 | nM |
Bosutinib | BTK | 4.80 | nM |
Bosutinib | M4K3 | 5.10 | nM |
Bosutinib | EPHA3 | 5.80 | nM |
Bosutinib | FGR | 6.30 | nM |
Bosutinib | LOK | 7.00 | nM |
Bosutinib | MP2K5 | 8.20 | nM |
Bosutinib | MAP4K4 | 8.20 | nM |
Bosutinib | EPHB2 | 8.40 | nM |
Bosutinib | EPHA8 | 9.00 | nM |
Bosutinib | EPHB4 | 9.20 | nM |
Bosutinib | MP2K2 | 9.90 | nM |
Bosutinib | FYN | 11.00 | nM |
Bosutinib | M4K1 | 15.00 | nM |
Bosutinib | YSK4 | 16.00 | nM |
Bosutinib | EPHA4 | 18.00 | nM |
Bosutinib | EGFR(E746-A750del) | 18.00 | nM |
Bosutinib | EPHA2 | 18.00 | nM |
Bosutinib | MP2K1 | 19.00 | nM |
Bosutinib | ABL1(T315I)-nonphosphorylated | 21.00 | nM |
Bosutinib | EGFR(L858R) | 23.00 | nM |
Bosutinib | ERBB4 | 26.00 | nM |