ABT-869 KINOMEscan - Dataset (ID:20182)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Linifanib | FES | nM | |
Linifanib | FGFR1 | nM | |
Linifanib | FGFR2 | nM | |
Linifanib | FGFR3 | nM | |
Linifanib | FGFR3(G697C) | nM | |
Linifanib | FGFR4 | nM | |
Linifanib | FGR | nM | |
Linifanib | VGFR1 | 7.5 | nM |
Linifanib | FLT3 | 0.6 | nM |
Linifanib | FLT3(D835H) | 2.7 | nM |
Linifanib | FLT3(D835Y) | 11.0 | nM |
Linifanib | FLT3(ITD) | 8.8 | nM |
Linifanib | FLT3(K663Q) | 1.3 | nM |
Linifanib | FLT3(N841I) | 2.6 | nM |
Linifanib | FLT3(R834Q) | 16.0 | nM |
Linifanib | FLT4 | 16.0 | nM |
Linifanib | FRK | 400.0 | nM |
Linifanib | FYN | nM | |
Linifanib | GAK | 2300.0 | nM |
Linifanib | GCN2(Kin.Dom.2,S808G) | nM | |
Linifanib | GRK1 | nM | |
Linifanib | GRK4 | nM | |
Linifanib | GRK7 | nM | |
Linifanib | GSK3A | nM | |
Linifanib | GSK3B | nM |