ABT-869 KINOMEscan - Dataset (ID:20182)

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Small Molecule Protein Kd Conc unit
Linifanib KIT 2.0
nM
Linifanib KIT(A829P) 17.0
nM
Linifanib KIT(D816H) 1100.0
nM
Linifanib KIT(D816V) 81.0
nM
Linifanib KIT(L576P) 1.9
nM
Linifanib KIT(V559D) 1.7
nM
Linifanib KIT(V559D,T670I) 3.8
nM
Linifanib KIT(V559D,V654A) 21.0
nM
Linifanib LATS1 2100.0
nM
Linifanib LATS2 1700.0
nM
Linifanib LCK
nM
Linifanib LIMK1
nM
Linifanib LIMK2 4700.0
nM
Linifanib LKB1
nM
Linifanib LOK 460.0
nM
Linifanib LRRK2
nM
Linifanib LRRK2(G2019S)
nM
Linifanib LTK 550.0
nM
Linifanib LYN
nM
Linifanib M3K13
nM
Linifanib MAK
nM
Linifanib MAP3K1
nM
Linifanib MAP3K15
nM
Linifanib M3K2
nM
Linifanib MAP3K3
nM