GDC-0879 KINOMEscan - Dataset (ID:20181)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| GDC-0879 | BRAF(V600E) | 0.2 | nM |
| GDC-0879 | BRAF | 0.2 | nM |
| GDC-0879 | RAF1 | 6.6 | nM |
| GDC-0879 | CSNK1E | 130.0 | nM |
| GDC-0879 | YSK4 | 910.0 | nM |
| GDC-0879 | MINK | 1000.0 | nM |
| GDC-0879 | RIOK2 | 1200.0 | nM |
| GDC-0879 | SLK | 1300.0 | nM |
| GDC-0879 | LOK | 1300.0 | nM |
| GDC-0879 | CSNK1D | 1400.0 | nM |
| GDC-0879 | BMPR1B | 1800.0 | nM |
| GDC-0879 | TNIK | 2300.0 | nM |
| GDC-0879 | MAP4K4 | 2300.0 | nM |
| GDC-0879 | ERBB3 | 2300.0 | nM |
| GDC-0879 | ACVR1B | 2400.0 | nM |
| GDC-0879 | RIPK2 | 2500.0 | nM |
| GDC-0879 | JNK3 | 2500.0 | nM |
| GDC-0879 | ABL1(H396P)-nonphosphorylated | 3200.0 | nM |
| GDC-0879 | CIT | 3500.0 | nM |
| GDC-0879 | TGFBR1 | 4900.0 | nM |
| GDC-0879 | MP2K5 | 5100.0 | nM |
| GDC-0879 | JAK1(JH2domain-pseudokinase) | 7800.0 | nM |
| GDC-0879 | ABL1-nonphosphorylated | nM | |
| GDC-0879 | ABL1(Y253F)-phosphorylated | nM | |
| GDC-0879 | ABL1(T315I)-phosphorylated | nM |